SCHEMBL11751680

SCHEMBL11751680

C/C(=N\C(C)C)c1cc2c(OCC(O)CNC(C)C)cccc2o1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 9/20 0.54
ADRB1 P08588 8/20 0.54
ADRB3 P13945 7/20 0.54
CYP1A2 P05177 5/20 0.54
CYP2D6 P10635 5/20 0.54
HTR1A P08908 5/20 0.54
SIGMAR1 Q99720 4/20 0.54
ALDH1A1 P00352 4/20 0.54
HTR2C P28335 4/20 0.54
LMNA P02545 4/20 0.54
SLC6A4 P31645 3/20 0.54
HTR2B P41595 3/20 0.54
NR2E1 Q9Y466 3/20 0.54
HTR2A P28223 3/20 0.54
HTR6 P50406 3/20 0.54
TSHR P16473 3/20 0.54
MAPK1 P28482 3/20 0.54
DRD3 P35462 3/20 0.54
SCN1A P35498 2/20 0.54
SLC10A1 Q14973 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11751687 1.00 ADRB2 (0.54) ADRB2ADRB1ADRB3CYP1A2CYP2D6
SCHEMBL11747691 0.84 ADRB2 (0.43) ADRB2ADRB1ADRB3CYP1A2CYP2D6
SCHEMBL11751411 0.83 ADRB2 (0.54) ADRB2ADRB1ADRB3CYP1A2CYP2D6
SCHEMBL11751418 0.83 ADRB2 (0.54) ADRB2ADRB1ADRB3CYP1A2CYP2D6
SCHEMBL11755136 0.78 ADRB2 (0.51) ADRB2ADRB1ADRB3CYP1A2CYP2D6
SCHEMBL11755128 0.78 ADRB2 (0.51) ADRB2ADRB1ADRB3CYP1A2CYP2D6
SCHEMBL11751694 0.75 ADRB2 (0.54) ADRB2ADRB1ADRB3CYP1A2CYP2D6
SCHEMBL10967303 0.73 LMNA (0.51) ADRB2ADRB1CYP1A2CYP2D6LMNA
SCHEMBL11748971 0.72 ADRB2 (0.64) ADRB2ADRB1ADRB3CYP1A2CYP2D6
SCHEMBL11868102 0.71 ADRB2 (0.82) ADRB2ADRB1ADRB3CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4056626-A ADRENERGIC BLOCKING AGENTS KAKENYAKU KAKO CO., LTD. (JA) 1977-11-01 US claimed
US-4056626-A ADRENERGIC BLOCKING AGENTS KAKENYAKU KAKO CO., LTD. (JA) 1977-11-01 US disclosed