SCHEMBL11763535

SCHEMBL11763535

COc1cc(Cc2c(N)nc(N)nc2O)cc(OC)c1OC

nearest known ligand 0.81

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.57
MEN1 O00255 1/20 0.57
SLC22A1 O15245 1/20 0.57
ALDH1A1 P00352 1/20 0.57
CYP3A4 P08684 1/20 0.57
TSHR P16473 1/20 0.57
NFKB1 P19838 1/20 0.57
CYP2C19 P33261 1/20 0.57
BLM P54132 1/20 0.57
KMT2A Q03164 1/20 0.57
HSD17B10 Q99714 1/20 0.57
SMN1; SMN2 Q16637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10681710 0.90 ALDH1A1 (0.48) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL11112703 0.87
SCHEMBL11112696 0.87 MEN1 (0.44) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL11166121 0.85 ALDH1A1 (0.43) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL11757871 0.84 DHFR (0.58) DHFRALDH1A1
SCHEMBL11345033 0.84 ALDH1A1 (0.43) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL11821666 0.83 DHFR (0.57) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL11859958 0.83 DHFR (0.43) DHFRALDH1A1
SCHEMBL15271540 0.79 DHFR (0.44) DHFRMEN1SLC22A1ALDH1A1CYP3A4
SCHEMBL12496384 0.78 HSP90AA1 (0.54) DHFRMEN1SLC22A1ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE29467-E Benzylcyano-amides PLANTEX, LTD. (IL) 1977-11-08 US disclosed
US-3980649-A Process for the manufacture of pyrimidine derivatives CHEMIE GRUNENTHAL GMBH (DT) 1976-09-14 US disclosed