SCHEMBL11166121

SCHEMBL11166121

COc1cc(Cc2c(N)nc(N)nc2O)cc(OC)c1SC

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
CYP2D6 P10635 1/20 0.43
ATM Q13315 1/20 0.43
MEN1 O00255 1/20 0.41
SLC22A1 O15245 1/20 0.41
DHFR P00374 1/20 0.41
CYP3A4 P08684 1/20 0.41
TSHR P16473 1/20 0.41
NFKB1 P19838 1/20 0.41
CYP2C19 P33261 1/20 0.41
BLM P54132 1/20 0.41
KMT2A Q03164 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10681710 0.86 ALDH1A1 (0.48) ALDH1A1CYP2D6ATMMEN1SLC22A1
SCHEMBL11763535 0.85 DHFR (0.57) ALDH1A1MEN1SLC22A1DHFRCYP3A4
SCHEMBL11166554 0.84 NPSR1 (0.44) ALDH1A1CYP2D6ATM
SCHEMBL11757871 0.81 DHFR (0.58) ALDH1A1CYP2D6ATMDHFR
SCHEMBL11345033 0.81 ALDH1A1 (0.43) ALDH1A1CYP2D6ATMMEN1SLC22A1
SCHEMBL11859958 0.80 DHFR (0.43) ALDH1A1CYP2D6ATMDHFR
SCHEMBL11112696 0.79 MEN1 (0.44) ALDH1A1MEN1SLC22A1DHFRCYP3A4
SCHEMBL11112703 0.79
Metioprim SCHEMBL193012 0.75 DHFR (0.73) ALDH1A1MEN1SLC22A1DHFRCYP3A4
Metioprim SCHEMBL30659007 0.75 DHFR (0.73) ALDH1A1MEN1SLC22A1DHFRCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0032395-B1 BENZYLPYRIMIDINES F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1983-03-23 EP disclosed
EP-0003212-B1 2.4-DIAMINO-5-BENZYLPYRIMIDINES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR PREPARATION F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1982-03-17 EP disclosed
EP-0032395-A1 Benzylpyrimidines F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1981-07-22 EP disclosed
EP-0003212-A1 2.4-Diamino-5-benzylpyrimidines, pharmaceutical compositions containing them and their preparation F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1979-08-08 EP disclosed