SCHEMBL11763585

SCHEMBL11763585

O=C(NC1CCCCC1)NS(=O)(=O)c1ccc2c(c1)CCN(C(=O)N1CCCC1)CC2

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.54
ALDH1A1 P00352 1/20 0.52
LMNA P02545 1/20 0.52
THRB P10828 1/20 0.52
TSHR P16473 1/20 0.52
BLM P54132 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
HRH3 Q9Y5N1 3/20 0.51
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
PPARG P37231 3/20 0.45
POLB P06746 1/20 0.45
HSD11B1 P28845 1/20 0.45
KCNA1 Q09470 5/20 0.44
KCNAB1 Q14722 5/20 0.44
MOGAT2 Q3SYC2 1/20 0.44
HPGD P15428 1/20 0.43
HTT P42858 1/20 0.43
NPC1 O15118 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11765186 1.00 ADORA3 (0.54) ADORA3ALDH1A1LMNATHRBTSHR
SCHEMBL11761408 0.92 ADORA3 (0.50) ADORA3ALDH1A1LMNATHRBTSHR
SCHEMBL11759176 0.89 ADORA3 (0.47) ADORA3ALDH1A1LMNATHRBTSHR
SCHEMBL11764729 0.87 ADORA3 (0.55) ADORA3ALDH1A1LMNATHRBTSHR
SCHEMBL11764048 0.87 KCNA1 (0.41) ADORA3ALDH1A1LMNATHRBTSHR
SCHEMBL11761600 0.86 ADORA3 (0.54) ADORA3ALDH1A1LMNATHRBTSHR
SCHEMBL11766631 0.86 ADORA3 (0.54) ADORA3ALDH1A1LMNATHRBTSHR
SCHEMBL11760402 0.86 ADORA3 (0.54) ADORA3ALDH1A1LMNATHRBTSHR
Glyhexamide SCHEMBL185244 0.86 ADORA3 (0.64) ADORA3ALDH1A1LMNATHRBTSHR
Glyhexamide SCHEMBL27491055 0.86 ADORA3 (0.64) ADORA3ALDH1A1LMNATHRBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4024128-A HYPOGLYCEMIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1977-05-17 US claimed
US-4024128-A HYPOGLYCEMIC AGENTS HOFFMANN-LA ROCHE INC. (US) 1977-05-17 US disclosed