SCHEMBL11782843

SCHEMBL11782843

COC(=O)C1CCCC(Br)C1=O

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
HIF1A Q16665 1/20 0.38
CHRM2 P08172 1/20 0.34
CHRM4 P08173 1/20 0.34
CHRM3 P20309 1/20 0.34
THRB P10828 1/20 0.33
BRD4 O60885 1/20 0.33
FKBP1A P62942 1/20 0.32
MAPK1 P28482 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TLR4 O00206 1/20 0.31
ALDH1A1 P00352 1/20 0.30
PPM1B O75688 1/20 0.30
PTPN1 P18031 1/20 0.30
KDM4E B2RXH2 1/20 0.30
HSD17B10 Q99714 1/20 0.30
PPP1CC P36873 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3362070 0.96 CYP1A2 (0.38) CYP1A2HIF1ACHRM2CHRM4CHRM3
SCHEMBL5514614 0.89 CYP1A2 (0.40) CYP1A2HIF1ATHRBBRD4ALDH1A1
SCHEMBL3974812 0.86 CYP1A2 (0.43) CYP1A2HIF1ACHRM2CHRM4CHRM3
SCHEMBL1617437 0.81 TLR4 (0.49) SMN1; SMN2TLR4ALDH1A1KDM4EHSD17B10
SCHEMBL12798508 0.79 CYP1A2 (0.39) CYP1A2HIF1ACHRM2CHRM4CHRM3
SCHEMBL3310290 0.79 CYP1A2 (0.39) CYP1A2HIF1ACHRM2CHRM4CHRM3
SCHEMBL14903874 0.79
SCHEMBL13882832 0.78 CYP1A2 (0.46) CYP1A2HIF1ABRD4SMN1; SMN2ALDH1A1
SCHEMBL11738399 0.76 MAPK1 (0.33) MAPK1
SCHEMBL14877461 0.75 GAA (0.37) MAPK1SMN1; SMN2TLR4ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3988444-A Novel thiazole derivatives as insecticides and acaricides ROUSSEL-UCLAF (FR) 1976-10-26 US disclosed
US-3948939-A 9-Acyl-1,2,3,4-tetrahydrocarbazole-3 and 4-carboxylic acids STERLING DRUG INC. (US) 1976-04-06 US disclosed
US-3932433-A ACRACIDES ROUSSEL-UCLAF (FR) 1976-01-13 US disclosed
US-3912757-A 1,2,3,4-Tetrahydrodibenzothiophene-1-carboxylates STERLING DRUG INC 1975-10-14 US disclosed