SCHEMBL11786229

SCHEMBL11786229

Cc1ccc(N2CCN(CCc3ccc4ccccc4n3)CC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.59
NPSR1 Q6W5P4 1/20 0.59
SLC6A4 P31645 4/20 0.57
KDM4E B2RXH2 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
NPC1 O15118 1/20 0.49
XBP1 P17861 1/20 0.49
RAB9A P51151 1/20 0.49
KLF5 Q13887 1/20 0.49
ADRA1D P25100 1/20 0.48
ADRA1A P35348 1/20 0.48
ADRA1B P35368 1/20 0.48
HTR1A P08908 4/20 0.47
DRD3 P35462 3/20 0.46
DRD2 P14416 2/20 0.46
SLC6A2 P23975 2/20 0.46
HRH3 Q9Y5N1 1/20 0.46
PDE10A Q9Y233 1/20 0.45
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11785894 0.89 DRD2 (0.56) HTR1ADRD3DRD2HTR2AHTR2C
SCHEMBL11785927 0.87 DRD3 (0.60) SLC6A4SMN1; SMN2HTR1ADRD3DRD2
SCHEMBL11785971 0.87 SLC6A2 (0.53) SLC6A4NPC1RAB9AADRA1DADRA1A
SCHEMBL8323715 0.87 SLC6A4 (0.54) MAPTNPSR1SLC6A4KDM4ESMN1; SMN2
Centhaquine SCHEMBL29751033 0.86 DRD3 (0.58) SLC6A4ADRA1DADRA1AADRA1BHTR1A
SCHEMBL11784050 0.86 DRD4 (0.53) MAPTNPSR1SLC6A4KDM4ESMN1; SMN2
SCHEMBL11784383 0.86 SLC6A2 (0.59) MAPTSLC6A4KDM4ESMN1; SMN2NPC1
Centhaquine SCHEMBL10029638 0.86 DRD3 (0.58) SLC6A4ADRA1DADRA1AADRA1BHTR1A
Centhaquine SCHEMBL29991817 0.86 DRD3 (0.58) SLC6A4ADRA1DADRA1AADRA1BHTR1A
Centhaquine SCHEMBL11788684 0.85 DRD3 (0.57) SLC6A4ADRA1DADRA1AADRA1BHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3983121-A 1-Substituted 4-(β-2-quinolylethyl)piperazines and 1,2,3,4-tetrahydroquinolyl-ethyl analogues thereof COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 1976-09-28 US claimed