SCHEMBL11794850

SCHEMBL11794850

CC(C)OC(=O)Nc1ccccn1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.58
RAB9A P51151 6/20 0.58
PKM P14618 2/20 0.58
POLB P06746 1/20 0.56
GAA P10253 2/20 0.54
ALDH1A1 P00352 3/20 0.54
LMNA P02545 1/20 0.54
SMN1; SMN2 Q16637 5/20 0.54
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
F2 P00734 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
PIM1 P11309 1/20 0.50
ADORA2A P29274 1/20 0.50
ADORA2B P29275 1/20 0.50
ADORA1 P30542 1/20 0.50
FLT3 P36888 1/20 0.50
PIM3 Q86V86 1/20 0.50
AURKB Q96GD4 1/20 0.50
TP53 P04637 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5246669 0.89 NPC1 (0.56) NPC1RAB9APKMPOLBGAA
SCHEMBL27850895 0.84 GAA (0.54) NPC1RAB9APKMPOLBGAA
SCHEMBL11539873 0.84 NPC1 (0.64) NPC1RAB9APKMPOLBGAA
SCHEMBL10914234 0.83 KDM4E (0.59) NPC1RAB9APKMPOLBGAA
SCHEMBL29655221 0.82 NPC1 (0.66) NPC1RAB9APKMPOLBGAA
SCHEMBL17266541 0.82 NPC1 (0.66) NPC1RAB9APKMPOLBGAA
SCHEMBL22793352 0.80 GAA (0.54) NPC1RAB9APKMPOLBGAA
SCHEMBL13588766 0.78 NPC1 (0.70) NPC1RAB9APKMPOLBGAA
SCHEMBL2666190 0.77 ALDH1A1 (0.71) NPC1RAB9APKMPOLBGAA
SCHEMBL9089971 0.77 RAB9A (0.63) NPC1RAB9APKMGAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023020518-A1 N-CYCLOPROPYLPYRIDO [4, 3-D] PYRIMIDIN-4-AMINE DERIVATIVES AND USES THEREOF JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2023-02-23 WO disclosed
US-10774053-B2 HIV protease inhibitors GILEAD SCIENCES, INC. (US) 2020-09-15 US disclosed
US-20190210978-A1 HIV PROTEASE INHIBITORS GILEAD SCIENCES, INC. (US) 2019-07-11 US disclosed
US-3938986-A ISOPROPYL N-PHENYLCARBAMATE OR ISOPROPYL N-(3-CHLOROPHENYL)CARBAMATE AND 4-CHLOROPHENYL N-METHYLCARBAMATE PPG INDUSTRIES, INC. (US) 1976-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10774053-B2 HIV protease inhibitors PRSS1, SERPINB1, FURIN NPC1 89/4885RAB9A 1131/4885PKM 1554/4885
US-20190210978-A1 HIV PROTEASE INHIBITORS PRSS1, SERPINB1, HPN NPC1 180/4885RAB9A 1421/4885PKM 2183/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.