SCHEMBL11801136

SCHEMBL11801136

O=C1c2cccc3cccc(c23)C(=O)N1CC=CO

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HEXA P06865 6/20 0.58
HEXB P07686 6/20 0.58
CYP1B1 Q16678 1/20 0.57
ALDH1A1 P00352 7/20 0.57
KDM4E B2RXH2 6/20 0.57
HPGD P15428 5/20 0.57
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
MAPT P10636 2/20 0.57
HSD17B10 Q99714 2/20 0.57
CYP1A2 P05177 2/20 0.57
AKR1B1 P15121 1/20 0.57
ALOX15 P16050 1/20 0.57
ERCC1 P07992 1/20 0.53
FEN1 P39748 1/20 0.53
ERCC4 Q92889 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
OGA O60502 1/20 0.53
SMN1; SMN2 Q16637 2/20 0.50
GAA P10253 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9064466 0.84 CASP3 (0.53) ALDH1A1KDM4EMAPTNPSR1RAB9A
SCHEMBL15485550 0.83 CYP1B1 (0.57) HEXAHEXBCYP1B1ALDH1A1KDM4E
SCHEMBL7319904 0.81 CYP1B1 (0.62) HEXAHEXBCYP1B1ALDH1A1KDM4E
SCHEMBL2539263 0.79 ALDH1A1 (0.63) HEXAHEXBCYP1B1ALDH1A1KDM4E
SCHEMBL11678307 0.77 HEXA (0.73) HEXAHEXBCYP1B1ALDH1A1KDM4E
SCHEMBL10262751 0.76 CYP1B1 (0.71) HEXAHEXBCYP1B1ALDH1A1KDM4E
SCHEMBL10690102 0.74 KDM4E (0.47) HEXAHEXBCYP1B1ALDH1A1KDM4E
SCHEMBL10690108 0.74 KDM4E (0.47) HEXAHEXBCYP1B1ALDH1A1KDM4E
SCHEMBL11667909 0.74 NPSR1 (0.47) HEXAHEXBCYP1B1ALDH1A1KDM4E
SCHEMBL4997995 0.74 HEXA (1.00) HEXAHEXBCYP1B1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4006238-A Use of 2-(hydroxyalkyl)-1H-benz[de]isoquinoline-1,3(2H)-diones as anti-allergy agents E. R. SQUIBB & SONS, INC. (US) 1977-02-01 US disclosed
US-4006238-A Use of 2-(hydroxyalkyl)-1H-benz[de]isoquinoline-1,3(2H)-diones as anti-allergy agents E. R. SQUIBB & SONS, INC. (US) 1977-02-01 US disclosed