SCHEMBL11838366

SCHEMBL11838366

c1cc(-c2cc(C3CC3)no2)ccn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.49
DRD4 P21917 1/20 0.49
DRD3 P35462 1/20 0.49
SCD O00767 3/20 0.45
SCD5 Q86SK9 2/20 0.45
QPCT Q16769 1/20 0.41
CYP2C19 P33261 3/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
CYP2C9 P11712 2/20 0.41
PTK2 Q05397 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
USP30 Q70CQ3 1/20 0.39
S1PR1 P21453 2/20 0.38
MCHR1 Q99705 1/20 0.38
MKNK1 Q9BUB5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11839633 0.81 SCD (0.44) DRD2DRD4DRD3SCDSCD5
SCHEMBL25338446 0.81 DRD2 (0.51) DRD2DRD4DRD3QPCTCHRNB2
SCHEMBL11841512 0.80 SCD (0.50) DRD2DRD4DRD3SCDSCD5
SCHEMBL21834025 0.79 DRD2 (0.47) DRD2DRD4DRD3QPCTCYP2C19
SCHEMBL21834029 0.79 MKNK1 (0.43) DRD2DRD4DRD3QPCTCHRNB2
SCHEMBL11848067 0.78 SCD5 (0.49) DRD2DRD4DRD3SCDSCD5
SCHEMBL4576107 0.77 DRD2 (0.48) DRD2DRD4DRD3QPCTCHRNB2
SCHEMBL28663908 0.76 RAB9A (0.53) DRD2DRD4DRD3SCDSCD5
SCHEMBL25339145 0.74 CXCR1 (0.48) DRD2DRD4DRD3QPCTNPC1
SCHEMBL11783495 0.74 RAB9A (0.54) DRD2DRD4DRD3CYP2C19CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3957805-A TREATMENT OF PAIN, MUSCLE SPASMS, ANXIETY, INFLAMMATION, OR TENSION AMERICAN CYANAMID COMPANY (US) 1976-05-18 US claimed
US-3997530-A ANALGESIC, ANTIPYRETIC AMERICAN CYANAMID COMPANY (US) 1976-12-14 US disclosed
US-3957805-A TREATMENT OF PAIN, MUSCLE SPASMS, ANXIETY, INFLAMMATION, OR TENSION AMERICAN CYANAMID COMPANY (US) 1976-05-18 US disclosed