SCHEMBL1187616

SCHEMBL1187616

OC(C(F)(F)F)C(Cl)(Cl)Cl

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.44
CETP P11597 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14784780 0.79 LMNA (0.35) LMNACETPALDH1A1HSD17B10
SCHEMBL6029543 0.79 LMNA (0.44) LMNA
SCHEMBL2262667 0.76 CETP (0.39) CETPALDH1A1HSD17B10
SCHEMBL1023713 0.76 LMNA (0.58) LMNA
SCHEMBL199 0.76 CETP (0.39) CETPALDH1A1HSD17B10
SCHEMBL2852867 0.76 CETP (0.39) CETPALDH1A1HSD17B10
Chloroform SCHEMBL5313122 0.74 ALDH1A1 (0.41) LMNACETPALDH1A1HSD17B10
Chloroform SCHEMBL6152248 0.74 ALDH1A1 (0.41) LMNACETPALDH1A1HSD17B10
SCHEMBL11204825 0.73 LMNA (0.32) LMNA
Water SCHEMBL17223739 0.72 CETP (0.37) CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190119462-A1 Porous Polymer Scaffolds, and Methods of Making and Using the Same THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2019-04-25 US claimed
EP-3468704-A1 POROUS POLYMER SCAFFOLDS, AND METHODS OF MAKING AND USING THE SAME The Regents of The University of California (US) 2019-04-17 EP claimed
WO-2017218565-A1 POROUS POLYMER SCAFFOLDS, AND METHODS OF MAKING AND USING THE SAME THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2017-12-21 WO claimed
US-8471006-B2 Coupling agents for peptide synthesis UNIVERSITY OF MASSACHUSETTS (US) 2013-06-25 US disclosed
US-20120277428-A1 NEW COUPLING AGENTS FOR PEPTIDE SYNTHESIS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2012-11-01 US disclosed
US-8217169-B2 Coupling agents for peptide synthesis UNIVERSITY OF MASSACHUSETTS (US) 2012-07-10 US disclosed
US-20110028720-A1 New Coupling Agents for Peptide Synthesis NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-02-03 US disclosed
US-7812158-B2 Coupling agents for peptide synthesis UNIVERSITY OF MASSACHUSETTS (US) 2010-10-12 US disclosed
EP-1687318-A4 NEW COUPLING AGENTS FOR PEPTIDE SYNTHESIS UNIV MASSACHUSETTS (US) 2009-01-07 EP disclosed
US-20070112196-A1 New coupling agents for peptide synthesis NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2007-05-17 US disclosed
CN-1898254-A New coupling agents for peptide synthesis UNIV MASSACHUSETTS (US) 2007-01-17 CN disclosed
EP-1687318-A2 NEW COUPLING AGENTS FOR PEPTIDE SYNTHESIS University of Massachusetts (US) 2006-08-09 EP disclosed
WO-2005042562-A2 NEW COUPLING AGENTS FOR PEPTIDE SYNTHESIS THE UNIVERSITY OF MASSACHUSETTS (US) 2005-05-12 WO disclosed
JP-2002371028-A METHOD FOR PRODUCING 3,3,3-TRIFLUORO-2-HYDROXYPROPIONIC ACID DERIVATIVE CENTRAL GLASS CO LTD 2002-12-26 JP disclosed
US-3994871-A Process for the manufacture of peptides containing cystine CIBA-GEIGY CORPORATION (US) 1976-11-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120277428-A1 NEW COUPLING AGENTS FOR PEPTIDE SYNTHESIS NGLY1, NPPA, VIP LMNA 4717/4885CETP 2404/4885ALDH1A1 4753/4885
US-20070112196-A1 New coupling agents for peptide synthesis NGLY1, NPPA, VIP LMNA 4649/4885CETP 2754/4885ALDH1A1 4756/4885
US-20110028720-A1 New Coupling Agents for Peptide Synthesis NGLY1, NPPA, VIP LMNA 4717/4885CETP 2404/4885ALDH1A1 4753/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.