SCHEMBL11879486

SCHEMBL11879486

CCOc1ccnc(CC(N)=S)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.45
POLB P06746 1/20 0.45
CYP3A4 P08684 2/20 0.44
LMNA P02545 2/20 0.44
TSHR P16473 2/20 0.44
KDM4E B2RXH2 1/20 0.44
TP53 P04637 1/20 0.39
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
PARP10 Q53GL7 1/20 0.38
PRSS1 P07477 1/20 0.38
PRSS2 P07478 1/20 0.38
PRSS3 P35030 1/20 0.38
PLAU P00749 1/20 0.37
MAPT P10636 3/20 0.37
ADRA2A P08913 2/20 0.37
NQO1 P15559 1/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11881287 0.85 NOS1 (0.54) CYP1A2POLBCYP3A4LMNATSHR
SCHEMBL17115680 0.79 KDM4E (0.44) CYP1A2LMNATSHRKDM4ENOS3
SCHEMBL5657197 0.78 NOTUM (0.48) CYP3A4LMNAKDM4ETP53NOS3
SCHEMBL12585924 0.77 NQO1 (0.46) CYP1A2POLBCYP3A4TSHRTP53
SCHEMBL15709664 0.76 NOS1 (0.44) CYP1A2TSHRKDM4ENOS1NOS2
SCHEMBL11877316 0.76 PLAU (0.49) CYP1A2POLBCYP3A4LMNATSHR
SCHEMBL14012773 0.75 NOS1 (0.41) CYP1A2POLBCYP3A4LMNATSHR
SCHEMBL3641525 0.74 NOS3 (0.43) CYP3A4TSHRKDM4ETP53NOS3
SCHEMBL30041354 0.74 KMT2A (0.38) CYP1A2LMNATSHRKDM4ENOS3
SCHEMBL30697969 0.71 NOS1 (0.36) CYP1A2LMNATSHRKDM4ENOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-3932641-A THIOACETAMIDES SMITHKLINE CORPORATION (US) 1976-01-13 US disclosed
US-3931162-A N-Aminomethyl heterocyclic thioacetamides SMITHKLINE CORPORATION (US) 1976-01-06 US disclosed