SCHEMBL5657197

SCHEMBL5657197

CCOc1ccnc(CO)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.48
S1PR1 P21453 1/20 0.44
S1PR3 Q99500 1/20 0.44
NOS1 P29475 2/20 0.43
NOS2 P35228 2/20 0.43
NOS3 P29474 1/20 0.43
NQO1 P15559 1/20 0.43
TP53 P04637 2/20 0.40
CYP3A4 P08684 1/20 0.40
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
KDM4E B2RXH2 1/20 0.38
CYP19A1 P11511 1/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
LTA4H P09960 1/20 0.37
NPC1 O15118 3/20 0.37
PKM P14618 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29380253 0.85 KMT2A (0.42) S1PR1S1PR3NOS1NOS2NOS3
SCHEMBL14012773 0.85 NOS1 (0.41) NOTUMNOS1NOS2NOS3NQO1
SCHEMBL9669619 0.85 KMT2A (0.42) S1PR1S1PR3NOS1NOS2NOS3
SCHEMBL26462412 0.84 NCF1 (0.46) NOTUMS1PR1S1PR3NOS1NOS2
SCHEMBL12585924 0.84 NQO1 (0.46) NOS1NOS2NOS3NQO1TP53
SCHEMBL2454070 0.84 CYP2D6 (0.46) CYP3A4ALDH1A1HPGDKMT2ACYP19A1
SCHEMBL245100 0.82 NOS2 (0.62) NOS1NOS2NOS3TP53ALDH1A1
SCHEMBL29694712 0.82 NOS2 (0.62) NOS1NOS2NOS3TP53ALDH1A1
SCHEMBL3641525 0.81 NOS3 (0.43) NOS1NOS2NOS3NQO1TP53
SCHEMBL23554280 0.80 NOS2 (0.44) NOS1NOS2NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12065409-B2 Analogs of 2-pralidoxime as antidotes against organophosphorus nerve agents University of Pittsburgh—of the Commonwealth System of Higher Education (US) 2024-08-20 US disclosed
CN-111655677-B Benzimidazole compounds as agrochemicals 瑞戴格作物保护公司 2024-05-03 CN disclosed
EP-3697771-B1 BENZIMIDAZOLE COMPOUNDS AS AGRICULTURAL CHEMICALS REDAG CROP PROT LTD (GB) 2022-04-06 EP disclosed
US-11241013-B2 Benzimidazole compounds as agricultural chemicals REDAG CROP PROT LTD (GB) 2022-02-08 US disclosed
US-11241013-B2 Benzimidazole compounds as agricultural chemicals REDAG CROP PROT LTD (GB) 2022-02-08 US disclosed
US-20210317084-A1 Analogs of 2-Pralidoxime as Antidotes Against Organophosphorus Nerve Agents UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION 2021-10-14 US disclosed
US-20210204547-A1 BENZIMIDAZOLE COMPOUNDS AS AGRICULTURAL CHEMICALS REDAG CROP PROT LTD (GB) 2021-07-08 US disclosed
US-20210204547-A1 BENZIMIDAZOLE COMPOUNDS AS AGRICULTURAL CHEMICALS REDAG CROP PROT LTD (GB) 2021-07-08 US disclosed
CN-111655677-A Benzimidazole compounds as agrochemicals 瑞戴格作物保护公司 2020-09-11 CN disclosed
EP-3697771-A1 BENZIMIDAZOLE COMPOUNDS AS AGRICULTURAL CHEMICALS Redag Crop Protection Ltd (GB) 2020-08-26 EP disclosed
WO-2020027905-A2 ANALOGS OF 2-PRALIDOXIME AS ANTIDOTES AGAINST ORGANOPHOSPHORUS NERVE AGENTS UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2020-02-06 WO disclosed
WO-2019077345-A1 BENZIMIDAZOLE COMPOUNDS AS AGRICULTURAL CHEMICALS REDAG CROP PROTECTION LTD (GB) 2019-04-25 WO disclosed
WO-2019077345-A1 BENZIMIDAZOLE COMPOUNDS AS AGRICULTURAL CHEMICALS REDAG CROP PROTECTION LTD (GB) 2019-04-25 WO disclosed
US-7262185-B2 Benzazepine derivative, process for producing the same, and use TAKEDA CHEMICAL INDUSTRIES LTD. (JP) 2007-08-28 US disclosed
US-20040235822-A1 Benzazepine derivative, process for producing the same, and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-11-25 US disclosed
EP-1422228-A1 BENZAZEPINE DERIVATIVE, PROCESS FOR PRODUCING THE SAME, AND USE Takeda Chemical Industries, Ltd. (JP) 2004-05-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210317084-A1 Analogs of 2-Pralidoxime as Antidotes Against Organophosphorus Nerve Agents ACHE, DDT, BCHE NOTUM 359/4885S1PR1 2634/4885S1PR3 2404/4885
US-12065409-B2 Analogs of 2-pralidoxime as antidotes against organophosphorus nerve agents ACHE, DDT, BCHE NOTUM 359/4885S1PR1 2634/4885S1PR3 2404/4885
US-11241013-B2 Benzimidazole compounds as agricultural chemicals CYP3A4, CYP2C8, CYP2E1 NOTUM 120/4885S1PR1 3978/4885S1PR3 3049/4885
US-20040235822-A1 Benzazepine derivative, process for producing the same, and use CYP1B1, CYP1A1, CYP2E1 NOTUM 555/4885S1PR1 647/4885S1PR3 1042/4885
US-20210204547-A1 BENZIMIDAZOLE COMPOUNDS AS AGRICULTURAL CHEMICALS CYP3A4, CYP2C8, CYP2E1 NOTUM 120/4885S1PR1 3978/4885S1PR3 3049/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.