SCHEMBL11903481

SCHEMBL11903481

FC(F)(F)Oc1ccc2nc(-c3ccccc3)[nH]c2c1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.72
RUNX1 Q01196 6/20 0.68
CBFB Q13951 3/20 0.68
KDM4E B2RXH2 4/20 0.68
ALDH1A1 P00352 4/20 0.68
HPGD P15428 4/20 0.68
NPC1 O15118 4/20 0.68
RAB9A P51151 4/20 0.68
TP53 P04637 3/20 0.68
SMN1; SMN2 Q16637 3/20 0.68
HSD17B10 Q99714 3/20 0.68
TSHR P16473 2/20 0.68
NFKB1 P19838 2/20 0.68
NFKB2 Q00653 2/20 0.68
RELA Q04206 2/20 0.68
NPBWR1 P48145 1/20 0.63
MAPT P10636 3/20 0.63
USP2 O75604 1/20 0.63
LMNA P02545 1/20 0.63
DGAT1 O75907 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11903477 0.89 TRPV1 (0.57) TRPV1RUNX1CBFBKDM4EALDH1A1
SCHEMBL11903468 0.87 TRPV1 (0.74) TRPV1RUNX1CBFBKDM4EALDH1A1
SCHEMBL11903447 0.86 TRPV1 (0.73) TRPV1RUNX1CBFBKDM4EALDH1A1
SCHEMBL11903498 0.86 TRPV1 (0.77) TRPV1RUNX1CBFBKDM4EALDH1A1
SCHEMBL11903652 0.86 TRPV1 (0.77) TRPV1RUNX1CBFBKDM4EALDH1A1
SCHEMBL11903458 0.85 CYP11B1 (0.64) TRPV1RUNX1CBFBKDM4EALDH1A1
SCHEMBL11903474 0.85 TRPV1 (0.71) TRPV1RUNX1CBFBKDM4EALDH1A1
SCHEMBL11903492 0.84 NPC1 (0.66) TRPV1RUNX1CBFBKDM4EALDH1A1
SCHEMBL11903519 0.83 TRPV1 (0.72) TRPV1RUNX1CBFBKDM4EALDH1A1
SCHEMBL22452568 0.82 KDM4E (0.66) TRPV1RUNX1CBFBKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293780-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making U.S. DEPARTMENT OF ENERGY (US) 2012-10-23 US disclosed
US-8293780-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making U.S. DEPARTMENT OF ENERGY (US) 2012-10-23 US disclosed
US-8242284-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making THE UNITED STATES OF AMERICA AS REPRESENTED BY THE UNITED STATES DEPARTMENT OF ENERGY (US) 2012-08-14 US disclosed
US-8242284-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making THE UNITED STATES OF AMERICA AS REPRESENTED BY THE UNITED STATES DEPARTMENT OF ENERGY (US) 2012-08-14 US disclosed