SCHEMBL11903491

SCHEMBL11903491

OCc1nc2cc(OC(F)(F)F)ccc2[nH]1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RHEB Q15382 2/20 0.50
RUNX1 Q01196 2/20 0.46
PDE10A Q9Y233 1/20 0.46
KDM4E B2RXH2 2/20 0.45
GAA P10253 2/20 0.45
KMT2A Q03164 1/20 0.45
TDP1 Q9NUW8 1/20 0.44
CBFB Q13951 3/20 0.40
TRPV1 Q8NER1 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
KIF11 P52732 1/20 0.40
IDO1 P14902 1/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
HDAC1 Q13547 2/20 0.39
HDAC2 Q92769 2/20 0.39
SCN10A Q9Y5Y9 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11903493 0.88 RUNX1 (0.58) RHEBRUNX1PDE10ATDP1CBFB
SCHEMBL23389133 0.85 PDE10A (0.46) RHEBRUNX1PDE10AKDM4EGAA
SCHEMBL10284435 0.85 DDAH1 (0.49) RUNX1PDE10AKDM4EGAAKMT2A
SCHEMBL19494108 0.85 KDM4E (0.45) RHEBRUNX1PDE10AKDM4EGAA
SCHEMBL25987878 0.83 PDE10A (0.50) RHEBRUNX1PDE10AKDM4EGAA
SCHEMBL11903503 0.83 PDE10A (0.50) RUNX1PDE10AKDM4EGAAKMT2A
SCHEMBL11904657 0.82 PDE10A (0.44) RHEBRUNX1PDE10AKDM4EGAA
SCHEMBL16189003 0.82 PKM (0.51) RUNX1PDE10AKDM4EGAAKMT2A
Hydrochloric Acid SCHEMBL11903446 0.81 GRIN1 (0.52) RUNX1PDE10AGAANPC1LMNA
Hydrochloric Acid SCHEMBL11903592 0.81 GAA (0.56) RUNX1PDE10AKDM4EGAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8293780-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making U.S. DEPARTMENT OF ENERGY (US) 2012-10-23 US disclosed
US-8242284-B1 Anti-cancer agents based on 6-trifluoromethoxybenzimidazole derivatives and method of making THE UNITED STATES OF AMERICA AS REPRESENTED BY THE UNITED STATES DEPARTMENT OF ENERGY (US) 2012-08-14 US disclosed