SCHEMBL11904598

SCHEMBL11904598

CC(C)(C)OC(=O)Nc1ccc2c(c1)C(N)CCS2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA9 Q16790 1/20 0.42
SIRT2 Q8IXJ6 3/20 0.38
SIRT1 Q96EB6 2/20 0.38
PSMB8 P28062 1/20 0.37
DGAT1 O75907 2/20 0.37
MAP4K4 O95819 1/20 0.37
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SLC10A2 Q12908 1/20 0.36
CYP17A1 P05093 1/20 0.36
MMP8 P22894 2/20 0.36
MMP3 P08254 1/20 0.36
ACHE P22303 1/20 0.36
BACE1 P56817 1/20 0.36
LEF1 Q9UJU2 1/20 0.36
MAPKAPK2 P49137 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22872917 0.77 NPC1 (0.47) CA12CA1CA9SIRT2SIRT1
SCHEMBL30831920 0.77 NPC1 (0.47) CA12CA1CA9SIRT2SIRT1
SCHEMBL11904012 0.73 VHL (0.49) CA12CA1CA9PSMB8CYP17A1
SCHEMBL7909165 0.72 MMP8 (0.44) CA12CA1CA9NPC1RAB9A
SCHEMBL17920282 0.71 DGAT1 (0.47) CA12CA1CA9SIRT2SIRT1
SCHEMBL31406453 0.71 CA12 (0.55) CA12CA1CA9SIRT2SIRT1
SCHEMBL14904889 0.71 NPC1 (0.47) CA12CA1CA9SIRT2SIRT1
SCHEMBL20809519 0.70 PYGL (0.47) CA12CA1CA9SIRT2SIRT1
SCHEMBL21788610 0.70 SIRT2 (0.61) CA12CA1CA9SIRT2SIRT1
SCHEMBL1115122 0.69 CA12 (0.47) CA12CA1CA9SIRT2SIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2487171-A1 Dihydrobenzopyran, thiochroman, tetrahydroquinoleine and tetrahydronaphthalene derivatives and their use in anti-cancer therapy Université de Liège (BE) 2012-08-15 EP disclosed