SCHEMBL11904869

SCHEMBL11904869

CCCCCC(=O)Nn1cnc2cncnc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.55
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
NPC1 O15118 1/20 0.40
GLA P06280 1/20 0.40
MAPK1 P28482 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
DEGS1 O15121 1/20 0.40
POLB P06746 1/20 0.40
HTT P42858 2/20 0.40
NCOA1 Q15788 1/20 0.40
NCOA3 Q9Y6Q9 1/20 0.40
RAB9A P51151 1/20 0.40
FDPS P14324 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36
MAPT P10636 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5196533 0.99 LMNA (0.57) LMNAHDAC1HDAC6NPC1GLA
SCHEMBL5492366 0.75 ALOX15 (0.64) LMNANPC1L3MBTL1POLBHTT
SCHEMBL5407957 0.70 LMNA (0.63) LMNANPC1L3MBTL1HTTHPGD
SCHEMBL10774226 0.70 FDPS (0.41) LMNAHDAC1HDAC6FDPSMEN1
SCHEMBL3691691 0.69 FDPS (0.48) LMNAHDAC1HDAC6NPC1MAPK1
SCHEMBL15741497 0.68 LMNA (0.56) LMNAGLADEGS1POLBHTT
SCHEMBL5041084 0.65 FDPS (0.37) LMNAHDAC1HDAC6MAPK1FDPS
SCHEMBL11061438 0.65 LMNA (0.50) LMNADEGS1POLBRAB9AMEN1
SCHEMBL11172485 0.65 FDPS (0.44) LMNAHDAC1HDAC6NPC1RAB9A
SCHEMBL10500165 0.65 FDPS (0.44) LMNAHDAC1HDAC6FDPSMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2486039-A1 PURINE DERIVATIVES USEFUL AS HSP90 INHIBITORS Sloan Kettering Institute For Cancer Research (US) 2012-08-15 EP disclosed