SCHEMBL1195261

SCHEMBL1195261

O=C(O)c1c(-c2ccccc2)ccc2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.57
KMT2A Q03164 4/20 0.57
ALDH1A1 P00352 3/20 0.57
HPGD P15428 3/20 0.57
KDM4E B2RXH2 2/20 0.57
HSD17B10 Q99714 2/20 0.57
CYP1A2 P05177 1/20 0.57
GLA P06280 1/20 0.57
CYP2C19 P33261 1/20 0.57
WDR5 P61964 1/20 0.48
METAP2 P50579 2/20 0.47
METAP1 P53582 1/20 0.47
LDHA P00338 1/20 0.47
NR4A1 P22736 1/20 0.47
NR4A2 P43354 1/20 0.47
NR4A3 Q92570 1/20 0.47
CDC25B P30305 1/20 0.46
MAPT P10636 2/20 0.45
HTT P42858 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1661024 0.90 HSD17B10 (0.63) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL6378389 0.90 MEN1 (0.50) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL4856686 0.89 MEN1 (0.49) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL28578355 0.88 KDM4E (0.49) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL27970017 0.88 METAP2 (0.53) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL10783912 0.86 CYP1A2 (0.55) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL722165 0.85 BCAT2 (0.47) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL28928988 0.85 MEN1 (0.46) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL10783918 0.85 MEN1 (0.57) MEN1KMT2AALDH1A1HPGDKDM4E
SCHEMBL8418459 0.84 KDM4E (0.56) MEN1KMT2AALDH1A1HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7291621-B2 Substituted biaryl amides C5a receptor modulators NEUROGEN CORPORATION (US) 2007-11-06 US claimed
US-20060178414-A1 Substituted biaryl amides as C5a receptor modulators NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2006-08-10 US claimed
EP-1487796-A4 SUBSTITUTED BIARYL AMIDES AS C5A RECEPTOR MODULATORS NEUROGEN CORP (US) 2005-11-16 EP claimed
EP-1487796-A1 SUBSTITUTED BIARYL AMIDES AS C5A RECEPTOR MODULATORS NEUROGEN CORPORATION (US) 2004-12-22 EP claimed
US-20040048913-A1 Substituted biaryl amides as C5a receptor modulators NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2004-03-11 US claimed
WO-2003082826-A1 SUBSTITUTED BIARYL AMIDES AS C5A RECEPTOR MODULATORS NEUROGEN CORPORATION (US) 2003-10-09 WO claimed
CN-119639276-A Ink composition, semiconductor nanoparticle-polymer composite prepared therefrom, electronic device, and display device 三星电子株式会社 2025-03-18 CN disclosed
EP-3898181-B1 PARALLELISED 3D LITHOGRAPHY USING MUTI-BEAM, MULTI-COLOUR LIGHT-INDUCED POLYMERISATION KARLSRUHER INST TECHNOLOGIE (DE) 2025-01-01 EP disclosed
EP-3898181-A1 PARALLELISED 3D LITHOGRAPHY USING MUTI-BEAM, MULTI-COLOUR LIGHT-INDUCED POLYMERISATION Karlsruher Institut für Technologie (DE) 2021-10-27 EP disclosed
CN-211463155-U Reaction device for producing and preparing phenyl naphthoate compound 武汉海昕药物研究有限公司 2020-09-11 CN disclosed
WO-2020126154-A1 PARALLELISED 3D LITHOGRAPHY USING MUTI-BEAM, MULTI-COLOUR LIGHT-INDUCED POLYMERISATION Karlsruher Institut für Technologie (DE) 2020-06-25 WO disclosed
CN-109665958-A A kind of method that ruthenium catalysis prepares polysubstituted 1- naphthoic acid class compound 广州大学 2019-04-23 CN disclosed
US-9217053-B2 Active ester resin, thermosetting resin composition, cured product of same, semiconductor encapsulation material, prepreg, circuit board, and build-up film DIC CORPORATION (JP) 2015-12-22 US disclosed
US-20050096358-A1 Substituted biaryl amides as C5A receptor modulators NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2005-05-05 US disclosed
EP-0439585-B1 IMMOBILISATION OF LIGANDS BY RADIO-DERIVATIZED POLYMERS MAG GEORG MAYRHOFER & CO OHG (AT) 1997-10-29 EP disclosed
US-5241103-A Dissolving 1,4-dihydroxy-2-arylnaphthoate containing a dimer by-product in an alcohol/water mixed solvent and isolation of 2-arylnaaphthoate by crystallization SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1993-08-31 US disclosed
US-5196478-A Polystyrene, assays EPIPHARM ALLERGIE-SERVICE GESELLSCHAFT M.B.H. (AT) 1993-03-23 US disclosed
US-5162570-A PROCESS FOR PRODUCING 1,4-DIHYDROXY-2-ARYLNAPHTHOATE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1992-11-10 US disclosed
EP-0439585-A1 IMMOBILISATION OF LIGANDS BY RADIO-DERIVATIZED POLYMERS. EPIPHARM ALLERGIE SERVICE (AT) 1991-08-07 EP disclosed
WO-1991002768-A1 IMMOBILISATION OF LIGANDS BY RADIO-DERIVATIZED POLYMERS EPIPHARM ALLERGIE-SERVICE GESELLSCHAFT M.B.H. (AT) 1991-03-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040048913-A1 Substituted biaryl amides as C5a receptor modulators C5AR1, C5AR2, C3AR1 MEN1 2253/4885KMT2A 4285/4885ALDH1A1 1494/4885
US-20050096358-A1 Substituted biaryl amides as C5A receptor modulators C5AR1, C5AR2, C3AR1 MEN1 2407/4885KMT2A 4155/4885ALDH1A1 1680/4885
US-20060178414-A1 Substituted biaryl amides as C5a receptor modulators C5AR1, C5AR2, C3AR1 MEN1 2407/4885KMT2A 4155/4885ALDH1A1 1680/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.