SCHEMBL119541

SCHEMBL119541

COC(=O)c1ccc(S(=O)(=O)NCc2ccccc2)c(F)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.54
POLB P06746 2/20 0.54
FABP4 P15090 2/20 0.52
KMT2A Q03164 2/20 0.51
ALDH1A1 P00352 4/20 0.49
CA12 O43570 1/20 0.49
CA9 Q16790 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
HPGD P15428 2/20 0.47
LMNA P02545 2/20 0.47
MAPT P10636 1/20 0.47
MEN1 O00255 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
KDM4E B2RXH2 1/20 0.47
GAA P10253 1/20 0.47
PKM P14618 1/20 0.47
CXCR4 P61073 1/20 0.47
CCR8 P51685 1/20 0.46
CYP1A2 P05177 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL108588 0.86 POLB (0.55) SMN1; SMN2POLBFABP4KMT2AALDH1A1
SCHEMBL119144 0.85 FABP4 (0.61) SMN1; SMN2POLBFABP4KMT2AALDH1A1
SCHEMBL119461 0.79 POLB (0.72) SMN1; SMN2POLBALDH1A1CA12CA9
SCHEMBL18423317 0.77 KDM4E (0.47) POLBKMT2AALDH1A1CA1CA2
SCHEMBL119469 0.76 KMT2A (0.66) SMN1; SMN2KMT2ACA12CA9LMNA
SCHEMBL975460 0.76 CA9 (0.73) SMN1; SMN2FABP4KMT2AALDH1A1CA12
SCHEMBL3850206 0.76 POLB (0.72) SMN1; SMN2POLBALDH1A1CA12CA9
SCHEMBL16709810 0.75 CA1 (0.52) SMN1; SMN2KMT2AALDH1A1CA1CA2
SCHEMBL119269 0.75 SMN1; SMN2 (0.64) SMN1; SMN2POLBKMT2AALDH1A1CA12
SCHEMBL119854 0.75 MAPT (0.64) SMN1; SMN2ALDH1A1HPGDLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2012-04-19 US disclosed
EP-2424517-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RaQualia Pharma Inc (JP) 2012-03-07 EP disclosed
WO-2010125831-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2010-11-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120094964-A1 SULFAMOYL BENZOIC ACID DERIVATIVES AS TRPM8 ANTAGONISTS TRPM8, TRPM5, TRPM6 SMN1; SMN2 1501/4885POLB 4630/4885FABP4 918/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.