SCHEMBL11954589

SCHEMBL11954589

NC(=S)c1cc(C(=O)I)cc(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.50
CES2 O00748 2/20 0.47
ALDH1A1 P00352 1/20 0.40
P2RX1 P51575 2/20 0.37
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ASH1L Q9NR48 1/20 0.36
GPR35 Q9HC97 1/20 0.36
NOTUM Q6P988 1/20 0.36
NFKB1 P19838 2/20 0.36
JUN P05412 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
CTSL P07711 1/20 0.35
CTSB P07858 1/20 0.35
ATF1 P18846 1/20 0.35
RXRA P19793 1/20 0.35
RXRB P28702 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11298235 0.85 GAA (0.53) GAACES2ALDH1A1ASH1LNOTUM
SCHEMBL627496 0.82 GAA (0.56) GAACES2ALDH1A1MAPTLMNA
SCHEMBL628459 0.78 ALDH1A1 (0.46) GAACES2ALDH1A1MAPTLMNA
SCHEMBL12128243 0.76 GAA (0.46) GAACES2ALDH1A1ASH1LCTSL
SCHEMBL12128276 0.74 CTSL (0.47) GAACES2ALDH1A1ASH1LCTSL
SCHEMBL1198001 0.74 NOTUM (0.53) GAACES2ALDH1A1ASH1LNOTUM
SCHEMBL3587775 0.74 GAA (0.49) GAACES2ALDH1A1MAPTASH1L
SCHEMBL11300330 0.72 GAA (0.44) GAACES2MAPTLMNAPOLB
SCHEMBL16283601 0.71 GAA (0.42) GAACES2ALDH1A1ASH1LCTSL
SCHEMBL628084 0.70 RXRA (0.43) GAAALDH1A1ASH1LNOTUMCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012099807-A1 OLEFIN CONTAINING NUCLEAR TRANSPORT MODULATORS AND USES THEREOF KARYOPHARM THERAPEUTICS, INC. (US) 2012-07-26 WO disclosed