SCHEMBL11980433

SCHEMBL11980433

Nc1nc(F)nc2[nH]c(Cc3ccccc3)nc12

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.46
MAPT P10636 2/20 0.43
PKM P14618 2/20 0.43
KDM4E B2RXH2 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
PNP P00491 1/20 0.42
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
RAB9A P51151 1/20 0.41
HTR6 P50406 2/20 0.40
KMT2A Q03164 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
LTB4R Q15722 1/20 0.40
GRIN1 Q05586 1/20 0.39
GRIN2B Q13224 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3923325 0.85 GAA (0.45) GAAMAPTPKMKDM4ETDP1
SCHEMBL870860 0.79 PI4KA (0.52) GAAMAPTPKMKDM4ETDP1
SCHEMBL26968483 0.78 ADORA3 (0.46) GAAMAPTPKMKDM4ETDP1
SCHEMBL24377312 0.77 MPO (0.41) GAAMAPTNPC1ALDH1A1RAB9A
SCHEMBL19996855 0.77 MPO (0.41) GAAMAPTNPC1ALDH1A1RAB9A
SCHEMBL1859066 0.77 POLB (0.53) GAAKDM4EALDH1A1KMT2A
SCHEMBL1669717 0.76 HSP90AA1 (0.45) PKMNPC1ALDH1A1RAB9AKMT2A
SCHEMBL4849398 0.75 HSP90AA1 (0.48) ALDH1A1KMT2A
SCHEMBL26968335 0.75 ADORA2A (0.51) ADORA3ADORA2AADORA2BADORA1
SCHEMBL16347480 0.72 CYP1A2 (0.49) MAPTKDM4ETDP1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9926321-B2 Hsp90 inhibitors SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2018-03-27 US disclosed
US-20160310497-A1 PURINE DERIVATIVES USEFUL AS HSP90 INHIBITORS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH 2016-10-27 US disclosed
US-20160264577-A1 HSP90 INHIBITORS SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH 2016-09-15 US disclosed
US-9346808-B2 Hsp90 inhibitors SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2016-05-24 US disclosed
US-9328114-B2 Hsp90 inhibitors SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2016-05-03 US disclosed
US-20120208806-A1 Hsp90 Inhibitors SLOAN-KETTERING INSTITUTE FOR CANCER RESEARCH (US) 2012-08-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160264577-A1 HSP90 INHIBITORS HSP90AB1, HSP90B1, HSP90AB2P GAA 310/4885MAPT 2557/4885PKM 2777/4885
US-20120208806-A1 Hsp90 Inhibitors HSP90B1, HSP90AB1, HSP90AB2P GAA 289/4885MAPT 2025/4885PKM 3530/4885
US-20160310497-A1 PURINE DERIVATIVES USEFUL AS HSP90 INHIBITORS XDH, HSP90B1, HSP90AA1 GAA 345/4885MAPT 3907/4885PKM 2268/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.