SCHEMBL11997802

SCHEMBL11997802

BCOc1ccccc1-c1ccc(NC(=O)OC(C)(C)C)cc1[N+](=O)[O-]

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
HTT P42858 2/20 0.40
SMN1; SMN2 Q16637 3/20 0.39
NPC1 O15118 4/20 0.38
RAB9A P51151 4/20 0.38
MAPK1 P28482 2/20 0.38
MEN1 O00255 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
AR P10275 2/20 0.38
PRMT1 Q99873 1/20 0.38
GBA1 P04062 1/20 0.38
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37
MMP9 P14780 1/20 0.37
MMP8 P22894 1/20 0.37
MMP13 P45452 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL398048 0.91 ALDH1A1 (0.48) ALDH1A1HTTSMN1; SMN2NPC1MEN1
SCHEMBL28370017 0.76 ALDH1A1 (0.61) ALDH1A1HTTSMN1; SMN2MEN1LMNA
SCHEMBL13832427 0.74 ALDH1A1 (0.69) ALDH1A1HTTSMN1; SMN2NPC1RAB9A
SCHEMBL7447972 0.74 ALDH1A1 (0.53) ALDH1A1HTTSMN1; SMN2NPC1RAB9A
SCHEMBL7448057 0.74 ALDH1A1 (0.48) ALDH1A1HTTSMN1; SMN2NPC1RAB9A
SCHEMBL1697905 0.74 RAB9A (0.61) ALDH1A1SMN1; SMN2NPC1RAB9AMAPK1
SCHEMBL395262 0.73 TDP1 (0.49) SMN1; SMN2NPC1RAB9AMEN1MAPT
SCHEMBL29790609 0.73 AR (0.55) ALDH1A1HTTSMN1; SMN2MAPK1LMNA
SCHEMBL1181321 0.73 MAPT (0.44) MEN1MAPTKMT2A
SCHEMBL9116516 0.73 ALDH1A1 (0.47) ALDH1A1HTTSMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2532650-A2 Modulators of ATP-binding cassette transporters Vertex Pharmaceuticals Incorporated (US) 2012-12-12 EP disclosed
EP-2530075-A2 Modulators of ATP-binding cassette transporters Vertex Pharmaceuticals Incorporated (US) 2012-12-05 EP disclosed
EP-2522659-A2 Modulators of ATP-binding cassette transporters Vertex Pharmaceuticals Incorporated (US) 2012-11-14 EP disclosed
EP-2502914-A2 Modulators of ATP-binding cassette transporters Vertex Pharmaceuticals Incorporated (US) 2012-09-26 EP disclosed
EP-2502913-A2 Modulators of ATP-binding cassette transporters Vertex Pharmaceuticals Incorporated (US) 2012-09-26 EP disclosed
EP-2502912-A2 Modulators of ATP-binding cassette transporters Vertex Pharmaceuticals Incorporated (US) 2012-09-26 EP disclosed
EP-2502902-A2 Modulators of ATP-binding cassette transporters Vertex Pharmaceuticals Incorporated (US) 2012-09-26 EP disclosed
EP-2502911-A2 Modulators of ATP-binding cassette transporters Vertex Pharmaceuticals Incorporated (US) 2012-09-26 EP disclosed
EP-2489659-A1 Modulators of ATP-binding cassette transporters Vertex Pharmaceuticals Incorporated (US) 2012-08-22 EP disclosed