SCHEMBL12002016

SCHEMBL12002016

CC(C)Cc1c(C(=O)O)c(C(=O)O)c(OCc2ccccc2)c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
USP2 O75604 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
GLRA1 P23415 1/20 0.43
KCNA2 P16389 1/20 0.42
KCNA5 P22460 1/20 0.42
KCNA1 Q09470 1/20 0.42
KDM4E B2RXH2 1/20 0.41
LMNA P02545 2/20 0.40
LTB4R Q15722 1/20 0.40
LTB4R2 Q9NPC1 1/20 0.40
HPGD P15428 1/20 0.40
NR4A1 P22736 1/20 0.39
NR4A2 P43354 1/20 0.39
NR4A3 Q92570 1/20 0.39
EDNRA P25101 1/20 0.39
KCNA3 P22001 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1590791 0.84 ALDH1A1 (0.52) ALDH1A1USP2TSHRHSD17B10KCNA2
SCHEMBL1974562 0.83 DHODH (0.44) ALDH1A1TSHRHSD17B10KDM4ELMNA
SCHEMBL14431116 0.83 ALDH1A1 (0.44) ALDH1A1USP2TSHRHSD17B10KCNA2
SCHEMBL9606562 0.82 KMT2A (0.38) ALDH1A1TSHRHSD17B10KDM4ELMNA
SCHEMBL1590125 0.82 EDNRA (0.52) ALDH1A1USP2TSHRHSD17B10GLRA1
SCHEMBL13177151 0.82 LTB4R (0.45) ALDH1A1USP2TSHRHSD17B10KCNA2
SCHEMBL1590143 0.80 ALDH1A1 (0.49) ALDH1A1USP2TSHRHSD17B10GLRA1
SCHEMBL1591366 0.80 KCNA3 (0.55) ALDH1A1USP2TSHRHSD17B10KCNA2
SCHEMBL12002194 0.78 ALDH1A1 (0.43) ALDH1A1USP2TSHRHSD17B10GLRA1
SCHEMBL1590385 0.78 ALDH1A1 (0.47) ALDH1A1USP2TSHRHSD17B10GLRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1979317-B1 BENZOISOINDOLE DERIVATIVES FOR THE TREATMENT OF PAIN GLAXO GROUP LTD (GB) 2012-08-22 EP disclosed
WO-2007088189-A1 BENZOISOINDOLE DERIVATIVES FOR THE TREATMENT OF PAIN GLAXO GROUP LIMITED (GB) 2007-08-09 WO disclosed