SCHEMBL1200237

SCHEMBL1200237

COc1ccc([Si](C)(C)Cl)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.55
CA2 P00918 2/20 0.55
CA7 P43166 2/20 0.55
CA9 Q16790 2/20 0.55
CA12 O43570 1/20 0.55
CA14 Q9ULX7 1/20 0.55
ACHE P22303 1/20 0.46
ALDH1A1 P00352 5/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
TDP1 Q9NUW8 4/20 0.44
MAPK1 P28482 4/20 0.44
KDM4E B2RXH2 2/20 0.42
MAPT P10636 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
NPC1 O15118 1/20 0.42
GAA P10253 1/20 0.42
THRB P10828 1/20 0.42
RECQL P46063 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5305926 0.85 CA1 (0.55) CA1CA2CA7CA9CA12
SCHEMBL13939389 0.84 CA1 (0.39) CA1CA2CA7CA9CA12
SCHEMBL12816764 0.82 CA1 (0.58) CA1CA2CA7CA9CA12
SCHEMBL1225152 0.82 CA1 (0.58) CA1CA2CA7CA9CA12
SCHEMBL10476909 0.81 CA1 (0.50) CA1CA2CA7CA9CA12
SCHEMBL705667 0.81 ALDH1A1 (0.36) ALDH1A1ESR1HPGD
SCHEMBL28701305 0.79 CA1 (0.61) CA1CA2CA7CA9CA12
SCHEMBL275937 0.79 CA1 (0.61) CA1CA2CA7CA9CA12
SCHEMBL19862402 0.79 CA1 (0.61) CA1CA2CA7CA9CA12
SCHEMBL22472159 0.78 CA1 (0.52) CA1CA2CA7CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2165377-B1 ORGANIC LIGHT-EMITTING DIODES CONTAINING CARBENE TRANSITION METAL COMPLEX EMITTERS AND AT LEAST ONE COMPOUND SELECTED FROM DISILYLCARBAZOLES, DISILYLDIBENZOFURANS, DISILYLDIBENZOTHIOPHENES, DISILYLDIBENZOPHOSPHOLES, DISILYLDIBENZOTHIOPHENE S-OXIDES AND DISILYLDIBENZOTHIOPHENE S,S-DIOXIDES UDC IRELAND LTD (IE) 2021-04-28 EP disclosed
US-10766982-B2 Cationic polymerization of olefins using green acids LEWIS STEWART P (US) 2020-09-08 US disclosed
EP-3345983-B1 COMPOUNDS CONTAINING AT LEAST ONE DISILYL COMPOUND SELECTED FROM DISILYLCARBAZOLES, DISILYLDIBENZOFURANS, DISILYLDIBENZOTHIOPHENES, DISILYLDIBENZOPHOSPHOLES, DISILYLDIBENZOTHIOPHENE S-OXIDES AND DISILYLDIBENZOTHIOPHENE S, S-DIOXIDES UDC IRELAND LTD (IE) 2020-08-26 EP disclosed
US-20190330395-A1 CATIONIC POLYMERIZATION OF OLEFINS USING GREEN ACIDS LEWIS STEWART P (US) 2019-10-31 US disclosed
EP-3345983-A1 COMPOUNDS CONTAINING AT LEAST ONE DISILYL COMPOUND SELECTED FROM DISILYLCARBAZOLES, DISILYLDIBENZOFURANS, DISILYLDIBENZOTHIOPHENES, DISILYLDIBENZOPHOSPHOLES, DISILYLDIBENZOTHIOPHENE S-OXIDES AND DISILYLDIBENZOTHIOPHENE S, S-DIOXIDES UDC Ireland Limited (IE) 2018-07-11 EP disclosed
US-9919300-B2 1-hexene production process SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2018-03-20 US disclosed
EP-2173834-B1 ORGANIC LIGHT-EMITTING DIODES COMPRISING AT LEAST ONE DISILYL COMPOUND SELECTED FROM DISILYLCARBAZOLES, DISILYLDIBENZOFURANS and DISILYLDIBENZOTHIOPHENES UDC IRELAND LTD (IE) 2018-02-14 EP disclosed
EP-2484685-B1 TRANSITION METAL COMPLEX, PREPARATION METHOD FOR SAID TRANSITION METAL COMPLEX, TRIMERIZATION CATALYST, PREPARATION METHOD FOR 1-HEXENE, PREPARATION METHOD FOR ETHYLENE POLYMER, SUBSTITUTED CYCLOPENTADIENE COMPOUND, AND PREPARATION METHOD FOR SAID SUBSTITUTED CYCLOPENTADIENE COMPOUND SUMITOMO CHEMICAL CO (JP) 2017-11-01 EP disclosed
US-20170036200-A1 1-HEXENE PRODUCTION PROCESS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2017-02-09 US disclosed
EP-2128897-B1 SILICON DIELECTRIC TREATING AGENT FOR USE AFTER ETCHING, PROCESS FOR PRODUCING SEMICONDUCTOR DEVICE, AND SEMICONDUCTOR DEVICE FUJITSU LTD (JP) 2015-05-06 EP disclosed
WO-2003100134-A1 ELECTROCHEMICAL METHOD FOR THE PRODUCTION OF ORGANOFUNCTIONAL SILANES Consortium für elektrochemische Industrie GmbH (DE) 2003-12-04 WO disclosed
EP-0363584-B1 Silylation method GEN ELECTRIC (US) 1994-09-14 EP disclosed
EP-0284873-B1 SILYLATION METHOD GENERAL ELECTRIC COMPANY (US) 1993-09-01 EP disclosed
US-4946921-A POLYSILICATE CONTAINING HYDROXYPHENYL GROUP TORAY SILICONE COMPANY LIMITED (JP) 1990-08-07 US disclosed
US-4925963-A Process for reduction of organosilicon halides ETHYL CORPORATION (US) 1990-05-15 US disclosed
EP-0363584-A2 Silylation method GENERAL ELECTRIC COMPANY (US) 1990-04-18 EP disclosed
US-4918197-A CATALYTIC REACTION BETWEEN AROMATIC ACYLHALIDE AND HALOGENATED POLYSILANE GENERAL ELECTRIC COMPANY (US) 1990-04-17 US disclosed
EP-0342648-A2 Alkali-soluble organopolysiloxane TORAY SILICONE COMPANY, LIMITED (JP) 1989-11-23 EP disclosed
EP-0284873-A2 Silylation method GENERAL ELECTRIC COMPANY (US) 1988-10-05 EP disclosed
US-4709054-A REACTION OF AROMATIC ACYL HALIDE AND HALOGENATED POLYSILANE, TRANSITION METAL CATALYST GENERAL ELECTRIC COMPANY (US) 1987-11-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170036200-A1 1-HEXENE PRODUCTION PROCESS AP1M1, HK1, CYC1 CA1 811/4885CA2 1484/4885CA7 2636/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.