SCHEMBL12031801

SCHEMBL12031801

CC1CCCN1C(=O)CNC(=O)c1ccccc1Cl

nearest known ligand 0.62

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.56
PREP P48147 9/20 0.54
FAP Q12884 5/20 0.54
DPP4 P27487 3/20 0.54
ALDH1A1 P00352 2/20 0.52
USP2 O75604 1/20 0.51
CHRM2 P08172 1/20 0.51
CHRM5 P08912 1/20 0.51
CHRM3 P20309 1/20 0.51
DPP8 Q6V1X1 1/20 0.51
DPP9 Q86TI2 1/20 0.51
CHRM1 P11229 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12949782 1.00 RAB9A (0.56) RAB9APREPFAPDPP4ALDH1A1
SCHEMBL13377307 0.85 PREP (0.51) PREPFAPDPP4DPP8DPP9
SCHEMBL8287722 0.85 TAS1R3 (0.50) PREPFAPDPP4DPP8DPP9
SCHEMBL8286847 0.84 RAB9A (0.55) RAB9APREPFAPDPP4ALDH1A1
SCHEMBL12031356 0.84 PREP (0.50) PREPFAPDPP4
SCHEMBL13377363 0.84 PREP (0.58) PREPFAPDPP4ALDH1A1DPP8
SCHEMBL13377308 0.84 PREP (0.50) PREPFAPDPP4DPP8DPP9
SCHEMBL12031885 0.83 KMT2A (0.58) RAB9APREPFAPALDH1A1DPP8
SCHEMBL12949796 0.80 PREP (0.45) PREPFAPDPP4ALDH1A1DPP8
SCHEMBL16381895 0.80 USP2 (0.49) RAB9APREPFAPDPP4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2399915-A1 Process and intermediates for the preparation of aspartic acetal caspase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-12-28 EP disclosed