SCHEMBL8287722

SCHEMBL8287722

Cc1cccc(C(=O)NCC(=O)N2CCCC2C)c1Cl

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.50
TAS1R1 Q7RTX1 1/20 0.50
TAS1R2 Q8TE23 1/20 0.50
PREP P48147 13/20 0.48
FAP Q12884 4/20 0.48
DPP4 P27487 2/20 0.48
DPP8 Q6V1X1 1/20 0.48
DPP9 Q86TI2 1/20 0.48
P2RX7 Q99572 2/20 0.46
HPGD P15428 1/20 0.44
DPP7 Q9UHL4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8287698 0.87 PREP (0.47) TAS1R3TAS1R1TAS1R2PREPFAP
SCHEMBL12031801 0.85 RAB9A (0.56) PREPFAPDPP4DPP8DPP9
SCHEMBL12949782 0.85 RAB9A (0.56) PREPFAPDPP4DPP8DPP9
SCHEMBL12949796 0.84 PREP (0.45) PREPFAPDPP4DPP8DPP9
SCHEMBL16381899 0.82 P2RX7 (0.46) PREPFAPDPP4DPP8DPP9
SCHEMBL12031723 0.81 RAB9A (0.51) TAS1R3TAS1R1TAS1R2P2RX7
SCHEMBL13377307 0.80 PREP (0.51) PREPFAPDPP4DPP8DPP9
SCHEMBL12031885 0.78 KMT2A (0.58) PREPFAPDPP8DPP9HPGD
SCHEMBL12949922 0.77 PREP (0.54) PREPFAPDPP4DPP8DPP9
SCHEMBL13377273 0.77 PREP (0.43) PREPFAPDPP4DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005085236-A2 CASPASE INHIBITORS AND USES THEREOF VERTEX PHARMACEUTICALS INCORPORATED (US) 2005-09-15 WO disclosed