SCHEMBL1208780

SCHEMBL1208780

COC(=O)C(N)(C(=O)OC(C)(C)C)c1ccc(Nc2cc(F)ccc2CN2C(=O)N(c3ccc(F)c(C(F)(F)F)c3)C(=O)C2(C)C)cc1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
AR P10275 12/20 0.46
CNR1 P21554 1/20 0.41
PPARG P37231 1/20 0.37
PPARD Q03181 1/20 0.37
PPARA Q07869 1/20 0.37
PGR P06401 1/20 0.36
IGF1R P08069 1/20 0.35
HDAC1 Q13547 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3535057 0.86 AR (0.50) ARCNR1PGRIGF1RHDAC1
SCHEMBL3526165 0.84 AR (0.52) ARCNR1PGRHDAC1
SCHEMBL3528150 0.83 AR (0.56) ARCNR1
SCHEMBL1206915 0.82 AR (0.47) ARCNR1PPARGPPARDPPARA
SCHEMBL1208782 0.82 AR (0.44) ARCNR1PGRIGF1R
SCHEMBL3527116 0.82 AR (0.54) ARCNR1PGRHDAC1
SCHEMBL1207317 0.82 AR (0.49) ARCNR1PGR
SCHEMBL3666698 0.81 AR (0.51) ARCNR1PGR
SCHEMBL1207342 0.81 AR (0.44) ARCNR1IGF1RHDAC1
SCHEMBL3527421 0.80 AR (0.49) ARCNR1IGF1RHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110046105-A1 Heterocycle-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising them and use thereof SANOFI-AVENTIS (FR) 2011-02-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110046105-A1 Heterocycle-substituted imidazolidine-2,4-diones, process for preparation thereof, medicaments comprising them and use thereof GIPR, DDC, PGC AR 1832/4885CNR1 660/4885PPARG 23/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.