SCHEMBL12132142

SCHEMBL12132142

COc1c(C(C)=O)c(OCOc2c3occc3c(OC)c3c(=O)cc(C)oc23)c(OC)c2occc12

nearest known ligand 0.67

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.67
CYP1A1 P04798 1/20 0.67
CYP1A2 P05177 1/20 0.67
CYP3A4 P08684 1/20 0.67
CYP2D6 P10635 1/20 0.67
HPGD P15428 1/20 0.67
PDE4A P27815 1/20 0.67
MAPK1 P28482 1/20 0.67
CYP2C19 P33261 1/20 0.67
SMN1; SMN2 Q16637 1/20 0.67
CYP1B1 Q16678 1/20 0.67
KCNA3 P22001 13/20 0.59
MAPT P10636 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13920847 0.84 KCNA3 (0.82) KCNA3
SCHEMBL13920848 0.82 CYP3A4 (0.81) ALDH1A1CYP1A1CYP1A2CYP3A4CYP2D6
Khellin SCHEMBL9655 0.81 CYP3A4 (1.00) ALDH1A1CYP1A1CYP1A2CYP3A4CYP2D6
Khellin SCHEMBL30839911 0.81 CYP3A4 (1.00) ALDH1A1CYP1A1CYP1A2CYP3A4CYP2D6
SCHEMBL12132138 0.81 CYP1A1 (0.76) ALDH1A1CYP1A1CYP1A2CYP3A4CYP2D6
SCHEMBL1344680 0.79 CYP3A4 (0.76) ALDH1A1CYP1A1CYP1A2CYP3A4CYP2D6
SCHEMBL12132140 0.78 KCNA3 (0.76) KCNA3
SCHEMBL10300860 0.78 CYP3A4 (0.74) ALDH1A1CYP1A1CYP1A2CYP3A4CYP2D6
SCHEMBL1345196 0.78 CYP3A4 (0.74) ALDH1A1CYP1A1CYP1A2CYP3A4CYP2D6
SCHEMBL13920849 0.77 CYP3A4 (0.81) ALDH1A1CYP1A1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8063093-B2 Derivatives of 5-(halo)alkanoyl-6-hydroxy- benozofuran, benzothiophene, or indole; autoimmune diseases; systemic lupus erythematosis, rheumatoid arthritis, multiple sclerosis and psoriasis, transplant rejection; antiproliferative, anticarcinogenic, antidiabetic, antiinflammatory and antiulcer agents HARVEY ANDREW J (AU) 2011-11-22 US disclosed
US-20080221194-A1 Novel Potassium channel Blockers and Uses Thereof HARVEY ANDREW J 2008-09-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080221194-A1 Novel Potassium channel Blockers and Uses Thereof KCNAB1, KCNB1, KCNMB1 ALDH1A1 982/4885CYP1A1 1790/4885CYP1A2 2450/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.