SCHEMBL12137709

SCHEMBL12137709

CS(=O)(=O)c1ccc(-c2nc(N)nc(N)c2-c2cccc(O)c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.47
PTGS2 P35354 1/20 0.46
SCD O00767 1/20 0.46
PIK3CA P42336 2/20 0.45
PIK3CB P42338 2/20 0.45
PIK3CG P48736 2/20 0.45
PIK3CD O00329 1/20 0.45
PIK3C2B O00750 1/20 0.45
PDXK O00764 1/20 0.45
GAK O14976 1/20 0.45
MAP3K7 O43318 1/20 0.45
RIPK2 O43353 1/20 0.45
PIP5K1C O60331 1/20 0.45
STK16 O75716 1/20 0.45
PIK3C2G O75747 1/20 0.45
PRKD3 O94806 1/20 0.45
OXSR1 O95747 1/20 0.45
LATS1 O95835 1/20 0.45
ABL1 P00519 1/20 0.45
EGFR P00533 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12137683 0.89 PTGS2 (0.46) DHFRPTGS2SCDPIK3CAPIK3CB
SCHEMBL27612333 0.83 ADORA1 (0.61) DHFRPIK3CAPIK3CBPIK3CGPIK3CD
SCHEMBL12137918 0.79 PTGS2 (0.54) DHFRPTGS2GHSR
SCHEMBL12135584 0.78 CA12 (0.46) DHFRPTGS2SCDPIK3CAMTOR
SCHEMBL12137707 0.78 HEXA (0.57) DHFRPIK3CAPIK3CBPIK3CGPIK3CD
SCHEMBL12138076 0.78 PIK3CG (0.50) DHFRPIK3CAPIK3CBPIK3CGPIK3CD
SCHEMBL27631682 0.77 ADORA1 (0.61) DHFRPIK3CAPIK3CBPIK3CGPIK3CD
SCHEMBL27631513 0.77 PIK3CG (0.59) DHFRPIK3CAPIK3CBPIK3CGPIK3CD
SCHEMBL12137855 0.76 DHFR (0.56) DHFRPIK3CAPIK3CBPIK3CGPIK3CD
SCHEMBL3452763 0.75 PTGS2 (0.56) DHFRPTGS2ADORA1ADORA2AGHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110281838-A1 5-ALKYNYL-PYRIMIDINES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-11-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110281838-A1 5-ALKYNYL-PYRIMIDINES MKI67, CCNA1, CCNT1 DHFR 11/4885PTGS2 2504/4885SCD 3564/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.