SCHEMBL12168148

SCHEMBL12168148

CC(=O)c1cc(C(=O)O)n[nH]1

nearest known ligand 0.59

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 16/20 0.59
DAO P14920 1/20 0.59
HCAR3 P49019 3/20 0.53
MAPK1 P28482 1/20 0.48
CYTH3 O43739 1/20 0.48
BTK Q06187 1/20 0.48
EPN1 Q9Y6I3 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12011328 0.87 MAPK1 (0.52) HCAR2DAOHCAR3MAPK1CYTH3
SCHEMBL70577 0.85 HCAR2 (0.59) HCAR2DAOHCAR3MAPK1CYTH3
SCHEMBL1815487 0.83 MAPK1 (0.48) HCAR2DAOHCAR3MAPK1
Hydrochloric Acid SCHEMBL7723258 0.83 HCAR2 (0.57) HCAR2DAOHCAR3MAPK1CYTH3
SCHEMBL19987833 0.83 HCAR2 (0.57) HCAR2DAOHCAR3MAPK1CYTH3
Water SCHEMBL1267709 0.83 HCAR2 (0.57) HCAR2DAOHCAR3MAPK1CYTH3
Hydrochloric Acid SCHEMBL11595364 0.83 HCAR2 (0.57) HCAR2DAOHCAR3MAPK1CYTH3
SCHEMBL28638090 0.83 HCAR2 (0.57) HCAR2DAOHCAR3MAPK1CYTH3
SCHEMBL13279353 0.82 MAPK1 (0.47) HCAR2DAOHCAR3MAPK1
Ammonia Solution, Strong SCHEMBL28463590 0.81 HCAR2 (0.55) HCAR2DAOHCAR3MAPK1CYTH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 118 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-121577799-A Method for determining 5-acetyl-1H-pyrazole-3-carboxylic acid related substances 江苏联环药业股份有限公司 2026-02-27 CN claimed
CN-118546091-A 5-Acetyl-1H-pyrazole-3-carboxylic acid and preparation method and application thereof 济南尚博医药股份有限公司 2024-08-27 CN claimed
CN-111138289-B Compound and process for synthesizing 5-acetyl-1H-pyrazole-3-carboxylic acid by using same 奥锐特药业(天津)有限公司 2022-08-30 CN claimed
CN-111138289-A Compound and process for synthesizing 5-acetyl-1H-pyrazole-3-carboxylic acid by using same 奥锐特药业(天津)有限公司 2020-05-12 CN claimed
CN-118546091-B 5-Acetyl-1H-pyrazole-3-carboxylic acid and preparation method and application thereof 济南尚博医药股份有限公司 2026-04-10 CN disclosed
CN-118546091-B 5-Acetyl-1H-pyrazole-3-carboxylic acid and preparation method and application thereof 济南尚博医药股份有限公司 2026-04-10 CN disclosed
CN-121673226-A Preparation method of drug intermediate 5-acetyl-1H-pyrazole-3-carboxylic acid and compound 湖北宇阳药业有限公司 2026-03-17 CN disclosed
CN-121673226-A Preparation method of drug intermediate 5-acetyl-1H-pyrazole-3-carboxylic acid and compound 湖北宇阳药业有限公司 2026-03-17 CN disclosed
CN-121577799-A Method for determining 5-acetyl-1H-pyrazole-3-carboxylic acid related substances 江苏联环药业股份有限公司 2026-02-27 CN disclosed
CN-121577799-A Method for determining 5-acetyl-1H-pyrazole-3-carboxylic acid related substances 江苏联环药业股份有限公司 2026-02-27 CN disclosed
CN-121577799-A Method for determining 5-acetyl-1H-pyrazole-3-carboxylic acid related substances 江苏联环药业股份有限公司 2026-02-27 CN disclosed
CN-120058672-A Halogenated pyridylcarboxylic acid ester derivative and application thereof 贵州医科大学 2025-05-30 CN disclosed
US-20140051708-A1 PYRAZOLYL-PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2014-02-20 US disclosed
US-20140045906-A1 NEPRILYSIN INHIBITORS THERAVANCE BIOPHARMA R&D IP, LLC 2014-02-13 US disclosed
US-20140045906-A1 NEPRILYSIN INHIBITORS THERAVANCE BIOPHARMA R&D IP, LLC 2014-02-13 US disclosed
WO-2014025891-A1 NEPRILYSIN INHIBITORS THERAVANCE, INC. (US) 2014-02-13 WO disclosed
WO-2014025891-A1 NEPRILYSIN INHIBITORS THERAVANCE, INC. (US) 2014-02-13 WO disclosed
WO-2012139930-A1 PYRAZOLYL-PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2012-10-18 WO disclosed
US-20120232052-A1 ARYL CARBOXAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC. (JP) 2012-09-13 US disclosed
US-20120232052-A1 ARYL CARBOXAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC. (JP) 2012-09-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140045906-A1 NEPRILYSIN INHIBITORS MME, REN, ACE HCAR2 658/4885DAO 1503/4885HCAR3 347/4885
US-20140051708-A1 PYRAZOLYL-PYRIMIDINE DERIVATIVES AS KINASE INHIBITORS MAP3K1, MAP3K20, MAP3K6 HCAR2 3486/4885DAO 3149/4885HCAR3 3249/4885
US-20120232052-A1 ARYL CARBOXAMIDE DERIVATIVES AS TTX-S BLOCKERS SCN1B, SCN1A, SCN2B HCAR2 308/4885DAO 1554/4885HCAR3 474/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.