SCHEMBL12187

SCHEMBL12187

CN(c1ccc(F)cc1)C1COCC2CCCCC21

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.42
DDB1 Q16531 1/20 0.37
CRBN Q96SW2 1/20 0.37
HSD11B1 P28845 1/20 0.32
KCNH2 Q12809 1/20 0.31
SSTR3 P32745 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10613 0.71 TRPA1 (0.39) TRPA1DDB1CRBN
SCHEMBL24230553 0.71 DDB1 (0.42) TRPA1DDB1CRBN
SCHEMBL10109530 0.68 ALDH1A1 (0.36)
SCHEMBL10388 0.68 DDB1 (0.36) TRPA1DDB1CRBN
SCHEMBL15013072 0.68 TRPA1 (0.49) TRPA1DDB1CRBNKCNH2
SCHEMBL2790916 0.67 DDB1 (0.49) TRPA1DDB1CRBNKCNH2
SCHEMBL11954688 0.67 TRPA1 (0.55) TRPA1DDB1CRBNHSD11B1KCNH2
SCHEMBL11967091 0.67 TRPA1 (0.55) TRPA1DDB1CRBNHSD11B1KCNH2
SCHEMBL15014118 0.65 DDB1 (0.44) TRPA1DDB1CRBNKCNH2
SCHEMBL5480634 0.65 DDB1 (0.50) TRPA1DDB1CRBNKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011043954-A1 NOVEL TRPA1 ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-04-14 WO disclosed