SCHEMBL12193293

SCHEMBL12193293

COC(=O)C(=O)N1CCCC1(C)C

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 6/20 0.33
USP2 O75604 1/20 0.33
TSHR P16473 1/20 0.32
NFKB1 P19838 1/20 0.32
CYP2C19 P33261 1/20 0.32
KDM5A P29375 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2006948 0.80 USP2 (0.31) USP2
SCHEMBL1159435 0.80 MAPT (0.41) CNR2TSHR
SCHEMBL14930639 0.80 USP2 (0.42) CNR2USP2TSHRNFKB1CYP2C19
SCHEMBL1159175 0.78 TSHR (0.38) CNR2TSHRNFKB1CYP2C19KDM5A
SCHEMBL27844146 0.75 CNR2 (0.36) CNR2TSHRNFKB1CYP2C19KDM5A
SCHEMBL7874674 0.75 FKBP1A (0.31)
SCHEMBL8669400 0.75 FKBP1A (0.33) USP2
SCHEMBL6429489 0.75 FKBP1A (0.31)
SCHEMBL1355575 0.73 TSHR (0.41) CNR2TSHRNFKB1CYP2C19KDM5A
SCHEMBL12155643 0.73 TSHR (0.36) CNR2TSHRNFKB1CYP2C19KDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2252611-B1 (DIHYDRO)PYRROLO[2,1-A]ISOQUINOLINES ORGANON NV (NL) 2011-10-05 EP disclosed
WO-2009098283-A1 (DIHYDRO)PYRROLO[2,1-A]ISOQUINOLINES N.V. ORGANON (NL) 2009-08-13 WO disclosed