Tramazoline

Tramazoline

SCHEMBL121944

c1cc2c(c(NC3=NCCN3)c1)CCCC2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.69
CYP2D6 P10635 2/20 0.69
CYP2C19 P33261 2/20 0.69
ADRA2A P08913 9/20 0.57
ADRA2B P18089 8/20 0.57
ADRA2C P18825 8/20 0.57
ADRA1A P35348 4/20 0.57
ADRA1D P25100 3/20 0.57
ADRA1B P35368 3/20 0.57
HTR1D P28221 1/20 0.51
HTR7 P34969 2/20 0.49
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
SLC22A1 O15245 1/20 0.48
SLC22A3 O75751 1/20 0.48
HTR1A P08908 1/20 0.48
CYP2C9 P11712 1/20 0.48
HRH2 P25021 1/20 0.48
OPRK1 P41145 1/20 0.48
HIF1A Q16665 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Tramazoline SCHEMBL121943 0.99 LMNA (0.68) LMNACYP2D6CYP2C19ADRA2AADRA2B
Tramazoline SCHEMBL29362958 0.99 LMNA (0.68) LMNACYP2D6CYP2C19ADRA2AADRA2B
Tramazoline SCHEMBL8378445 0.97 LMNA (0.67) LMNACYP2D6CYP2C19ADRA2AADRA2B
Indanazoline SCHEMBL151815 0.97 LMNA (0.66) LMNACYP2D6CYP2C19ADRA2AADRA2B
Indanazoline SCHEMBL1650054 0.96 LMNA (0.65) LMNACYP2D6CYP2C19ADRA2AADRA2B
Indanazoline SCHEMBL3500123 0.96 LMNA (0.65) LMNACYP2D6CYP2C19ADRA2AADRA2B
Tramazoline SCHEMBL4760046 0.88 LMNA (0.63) LMNACYP2D6CYP2C19ADRA2AADRA2B
Indanazoline SCHEMBL11372740 0.87 LMNA (0.66) LMNACYP2D6CYP2C19ADRA2AADRA2B
Tramazoline SCHEMBL28086399 0.81 TAAR1 (0.61) LMNACYP2D6CYP2C19ADRA2AADRA2B
Indanazoline SCHEMBL3064466 0.81 ADRA1A (0.67) LMNACYP2D6CYP2C19ADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4548 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-122075410-A Dry powder composition for intranasal delivery 2026-05-26 CN claimed
US-20260108531-A1 Methods of Treating Hypogonadism with Transnasal Testosterone Bio-adhesive Gel Formulations in Males with Allergic Rhinitis and Methods for Preventing an Allergic Rhinitis Event ACERUS BIOPHARMA INC (CA) 2026-04-23 US claimed
US-12605345-B2 Transdermal drug delivery system BioPhysics Pharma, Inc. (US) 2026-04-21 US claimed
CN-120114603-A Compound pharmaceutical composition for treating presbyopia as well as preparation method, application and preparation thereof 立生医药(苏州)有限公司 2025-06-10 CN claimed
EP-3359134-B1 COMPOSITIONS AND COMPOSITIONS FOR USE IN ON-DEMAND HIGH-EFFICIENCY TRIGGERABLE ANESTHESIA CHILDRENS MEDICAL CT CORP (US) 2025-04-09 EP claimed
CN-119700672-A An eye spray composition for relieving ptosis and redeye 立生医药(苏州)有限公司 2025-03-28 CN claimed
US-20250049761-A1 COMPOSITIONS AND METHODS FOR TREATING PRESBYOPIA, MILD HYPEROPIA, AND IRREGULAR ASTIGMATISM ALLERGAN, INC. 2025-02-13 US claimed
US-20240316063-A1 METHODS OF TREATING HYPOGONADISM WITH TRANSNASAL TESTOSTERONE BIO-ADHESIVE GEL FORMULATIONS IN MALE WITH ALLERGIC RHINITIS, AND METHODS FOR PREVENTING AN ALLERGIC RHINITIS EVENT ACERUS BIOPHARMA INC (CA) 2024-09-26 US claimed
EP-3756665-B1 INTERVAL THERAPY FOR THE TREATMENT OF EYE DISEASES UNIV RAMOT (IL) 2024-08-14 EP claimed
US-20240108588-A1 Transdermal Drug Delivery System Masiz, John J. (US) 2024-04-04 US claimed
WO-1993024149-A1 PHARMACEUTICAL POWDER COMPOSITION CONTAINING NON-IONIC CELLULOSE ETHER DERIVATIVE AND A CHITIN-DERIVED POLYMER THE PROCTER & GAMBLE COMPANY (US) 1993-12-09 WO claimed
EP-0571671-A1 A Pharmaceutical composition in powder form THE PROCTER & GAMBLE COMPANY (US) 1993-12-01 EP claimed
EP-0550921-A1 Pharmaceutical composition for ophthalmic use comprising a nonsteroidal anti-inflammatory and a decongestant drug ZAMBON GROUP S.p.A. (IT) 1993-07-14 EP claimed
WO-1992014453-A1 COMPOSITIONS AND METHODS OF TREATMENT OF SYMPATHETICALLY MAINTAINED PAIN ARC 1, INC. (US) 1992-09-03 WO claimed
EP-0170193-B1 FEEDSTUFF ADDITIVE FOR THE GROWTH PROMOTING OF AGRICULTURAL USEFUL ANIMALS BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 1991-12-27 EP claimed
EP-0448299-A2 Composition for increased skin concentration of active agents by iontophoresis Becton, Dickinson and Company (US) 1991-09-25 EP claimed
US-4853402-A 2-SUBSTITUTED-2-IMIDAZOLINES BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 1989-08-01 US claimed
EP-0086428-B1 ANTIDIARRHOEA VETERINARY COMPOSITION, ITS PRODUCTION AND ORAL DOSER CONTAINING IT BEECHAM GROUP PLC (GB) 1987-07-29 EP claimed
EP-0170193-A2 Feedstuff additive for the growth promoting of agricultural useful animals BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 1986-02-05 EP claimed
EP-0025269-B1 ANTI-DIARRHOEA VETERINARY COMPOSITION BEECHAM GROUP PLC (GB) 1985-11-13 EP claimed