SCHEMBL12200364

SCHEMBL12200364

Nc1ccc(C(=O)NC2CCNCC2)cc1Cl

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 1/20 0.57
SMYD3 Q9H7B4 6/20 0.53
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
KHK P50053 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
CHEK1 O14757 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
UTS2R Q9UKP6 2/20 0.45
CCNT1 O60563 1/20 0.44
CDK9 P50750 1/20 0.44
CDK5 Q00535 1/20 0.44
CDK5R1 Q15078 1/20 0.44
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6824779 0.87 SMYD3 (0.56) SMYD3MEN1KMT2AUTS2RHDAC8
SCHEMBL13575477 0.83 HDAC6 (0.55) HTR4SMYD3KHKNPC1RAB9A
SCHEMBL13575614 0.83 SMYD3 (0.53) HTR4SMYD3MEN1KMT2AKHK
SCHEMBL1711760 0.83 TAS1R3 (0.57) SMYD3MEN1KMT2AKHKL3MBTL1
SCHEMBL10144490 0.81 HTR4 (0.61) HTR4SMYD3MEN1KMT2AKHK
SCHEMBL1559555 0.81 KMT2A (0.49) HTR4SMYD3MEN1KMT2AUTS2R
SCHEMBL13575615 0.81 SMYD3 (0.51) HTR4SMYD3KMT2AKHKNPC1
SCHEMBL13575536 0.80 TAS1R3 (0.54) HTR4SMYD3KHKHDAC3HDAC4
SCHEMBL10078319 0.80 HTR4 (0.60) HTR4SMYD3
SCHEMBL13575468 0.79 KHK (0.54) SMYD3MEN1KMT2AKHKNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2135608-B1 S-triazolyl alpha -mercaptoacetanilides as inhibitors of HIV reverse transcriptase ARDEA BIOSCIENCES INC (US) 2011-10-12 EP disclosed