SCHEMBL13575615

SCHEMBL13575615

CCc1cc(C(=O)NC2CCNCC2)ccc1N

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 8/20 0.51
KHK P50053 4/20 0.47
HTR4 Q13639 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
HDAC9 Q9UKV0 1/20 0.46
HDAC5 Q9UQL6 1/20 0.46
ACSS2 Q9NR19 1/20 0.45
NPC1 O15118 2/20 0.44
MAPK14 Q16539 1/20 0.43
HPGDS O60760 1/20 0.43
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13575588 0.84 KDM1A (0.54) SMYD3ACSS2NPC1RAB9AKMT2A
SCHEMBL13575614 0.84 SMYD3 (0.53) SMYD3KHKHTR4HDAC3HDAC4
SCHEMBL4052654 0.83 ACSS2 (0.47) SMYD3HDAC4HDAC6ACSS2NPC1
SCHEMBL13575620 0.83 HPGD (0.51) SMYD3KHKHTR4HPGDSRAB9A
SCHEMBL13575520 0.82 HTR4 (0.52) SMYD3HTR4NPC1HPGDSRAB9A
SCHEMBL10144490 0.82 HTR4 (0.61) SMYD3KHKHTR4HPGDSKMT2A
SCHEMBL12200364 0.81 HTR4 (0.57) SMYD3KHKHTR4HDAC3HDAC4
SCHEMBL13575477 0.81 HDAC6 (0.55) SMYD3KHKHTR4HDAC3HDAC4
SCHEMBL13880649 0.79 MAPK1 (0.58) SMYD3KHKHTR4HPGDSKMT2A
SCHEMBL13575536 0.78 TAS1R3 (0.54) SMYD3KHKHTR4HDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009153197-A1 HALO-SUBSTITUTED PYRIMIDODIAZEPINES AS PLKL INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2009-12-23 WO disclosed