SCHEMBL12209643

SCHEMBL12209643

CN1CCC(N(C)C(=O)c2cccc(C3CCNCC3)c2)CC1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 7/20 0.44
MAPT P10636 1/20 0.43
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
TLR9 Q9NR96 1/20 0.42
TLR8 Q9NR97 1/20 0.42
TLR7 Q9NYK1 1/20 0.42
CCR5 P51681 1/20 0.42
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
HTR2A P28223 1/20 0.40
KDM4E B2RXH2 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8054566 0.90 HTR2C (0.50) HTR2CALDH1A1POLBKDM4EHPGD
SCHEMBL8054636 0.85 MCHR1 (0.45) LMNATLR9TLR8TLR7CCR5
SCHEMBL12209651 0.85 HTR2C (0.45) HTR2CALDH1A1POLBKDM4EHPGD
SCHEMBL30804745 0.79 KMT2A (0.59) HTR2CMAPTALDH1A1LMNAPOLB
SCHEMBL16488097 0.78 QDPR (0.46) ALDH1A1LMNAPOLBL3MBTL1KMO
SCHEMBL3329900 0.77 CCR5 (0.55) HTR2CPOLBADORA2AADORA1CCR5
SCHEMBL30804735 0.76 MCHR1 (0.53) MAPTALDH1A1POLBL3MBTL1
SCHEMBL30804752 0.76 MCHR1 (0.53) MAPTALDH1A1POLBL3MBTL1
SCHEMBL13609464 0.75 HCRTR1 (0.56) HTR2CALDH1A1LMNAHPGD
SCHEMBL373768 0.74 LIMK2 (0.47) HTR2CALDH1A1POLBL3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2380891-A1 Substituted piperidino-dihydrothienopyrimidines BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-10-26 EP disclosed