SCHEMBL12246

SCHEMBL12246

C=C1N(c2ccc(CC(C)C)cc2)CC[C@]12CC[C@@](O)(C(C)C)CC2

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 5/20 0.34
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
OPRL1 P41146 1/20 0.33
MMP1 P03956 1/20 0.32
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32
ADAM17 P78536 1/20 0.32
TSHR P16473 1/20 0.32
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12117 0.85 LIPE (0.33) LIPEMMP1MMP2MMP9ADAM17
SCHEMBL5254 0.69 LIPE (0.48) LIPE
SCHEMBL1589517 0.65 LIPE (0.58) LIPE
SCHEMBL1589513 0.65 LIPE (0.58) LIPE
SCHEMBL10124 0.65 LIPE (0.65) LIPE
SCHEMBL10123 0.65 LIPE (0.65) LIPE
SCHEMBL12193 0.64 MCOLN3 (0.40) LIPEMEN1KMT2AL3MBTL1
SCHEMBL12702001 0.63 LIPE (0.69) LIPE
SCHEMBL11778 0.63 LIPE (0.62) LIPE
SCHEMBL12702172 0.63 LIPE (0.62) LIPE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011045292-A1 SPIRO-CONDENSED CYCLOHEXANE DERIVATIVES AS HSL INHIBITORS USEFUL FOR THE TREATMENT OF DIABETES F. HOFFMANN-LA ROCHE AG (CH) 2011-04-21 WO disclosed