SCHEMBL12193

SCHEMBL12193

C=C1N(c2ccc(C(C)C)cc2)CCC12CCC(C)CC2

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MCOLN3 Q8TDD5 1/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
HPGD P15428 1/20 0.36
HRH3 Q9Y5N1 6/20 0.34
LIPE Q05469 3/20 0.34
HSD11B1 P28845 1/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
MGLL Q99685 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12346 0.79 POLB (0.32) LIPEMEN1KMT2ACYP1A2CYP2C9
SCHEMBL12024 0.78 LIPE (0.35) LIPE
SCHEMBL10832 0.70 HRH3 (0.52) HRH3LIPEHSD11B1
SCHEMBL12701963 0.70 HRH3 (0.52) HRH3LIPEHSD11B1
SCHEMBL5672 0.70 HRH3 (0.52) HRH3LIPEHSD11B1
SCHEMBL10147276 0.70 USP2 (0.54) MCOLN3L3MBTL1HPGDHRH3HSD11B1
SCHEMBL9601 0.67 LIPE (0.42) L3MBTL1LIPEHSD11B1MEN1KMT2A
SCHEMBL4438936 0.65 MCOLN3 (0.41) MCOLN3L3MBTL1HPGDHSD11B1
SCHEMBL16786535 0.65 MGLL (0.45) L3MBTL1HPGDMEN1KMT2ACYP1A2
SCHEMBL24720951 0.65 RAB9A (0.50) L3MBTL1LIPEHSD11B1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011045292-A1 SPIRO-CONDENSED CYCLOHEXANE DERIVATIVES AS HSL INHIBITORS USEFUL FOR THE TREATMENT OF DIABETES F. HOFFMANN-LA ROCHE AG (CH) 2011-04-21 WO disclosed