SCHEMBL12117

SCHEMBL12117

C=C(C)[C@]1(O)CC[C@]2(CCN(c3ccc(CC(C)C)cc3)C2=C)CC1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 4/20 0.33
MMP1 P03956 1/20 0.31
MMP2 P08253 1/20 0.31
MMP9 P14780 1/20 0.31
ADAM17 P78536 1/20 0.31
TSHR P16473 1/20 0.30
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12346 0.84 POLB (0.32) LIPEMEN1POLBKMT2A
SCHEMBL1589420 0.71 LIPE (0.43) LIPE
SCHEMBL11103 0.69 LIPE (0.45) LIPE
SCHEMBL11972 0.64 LIPE (0.52) LIPE
SCHEMBL20684172 0.63 SMN1; SMN2 (0.43) TSHRMEN1NPC1ALDH1A1POLB
SCHEMBL12193 0.63 MCOLN3 (0.40) LIPEMEN1KMT2AL3MBTL1
SCHEMBL12336 0.62 TRPV1 (0.33) LIPE
SCHEMBL8244253 0.59 CHKA (0.46) TSHRMEN1NPC1ALDH1A1POLB
SCHEMBL17897210 0.58 ACACB (0.55) TSHRMEN1ALDH1A1KMT2A
SCHEMBL4669161 0.58 PTGS1 (0.46) TSHRMEN1ALDH1A1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011045292-A1 SPIRO-CONDENSED CYCLOHEXANE DERIVATIVES AS HSL INHIBITORS USEFUL FOR THE TREATMENT OF DIABETES F. HOFFMANN-LA ROCHE AG (CH) 2011-04-21 WO disclosed