SCHEMBL12264154

SCHEMBL12264154

OC(c1ccccc1)(c1ccccc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.71
ALDH1A1 P00352 1/20 0.70
TSHR P16473 1/20 0.70
KIF11 P52732 2/20 0.58
TRPV6 Q9H1D0 2/20 0.54
CYP3A4 P08684 3/20 0.50
CYP2D6 P10635 1/20 0.50
CYP3A5 P20815 2/20 0.49
RAB9A P51151 2/20 0.47
NPC1 O15118 1/20 0.47
AHR P35869 1/20 0.46
ACP3 P15309 1/20 0.46
USP2 O75604 1/20 0.45
CES2 O00748 1/20 0.44
CES1 P23141 1/20 0.44
ORAI1 Q96D31 1/20 0.44
ORAI2 Q96SN7 1/20 0.44
ORAI3 Q9BRQ5 1/20 0.44
MGLL Q99685 1/20 0.44
BACE1 P56817 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9050608 0.87 CYP19A1 (0.54) CYP19A1ALDH1A1TSHRCYP3A4CYP2D6
SCHEMBL30915210 0.85 ALDH1A1 (0.70) CYP19A1ALDH1A1TSHRKIF11TRPV6
SCHEMBL7766770 0.85 ALDH1A1 (0.70) CYP19A1ALDH1A1TSHRKIF11TRPV6
SCHEMBL12264155 0.84 CYP19A1 (0.55) CYP19A1ALDH1A1TSHRKIF11CYP3A4
Triphenylmethanol SCHEMBL1332873 0.84 CYP19A1 (0.50) CYP19A1ALDH1A1TSHRCYP3A4CYP2D6
Trifluoromethylbenzene SCHEMBL27760126 0.84 TSHR (1.00) CYP19A1ALDH1A1TSHRKIF11TRPV6
Trifluoromethylbenzene SCHEMBL175647 0.84 TSHR (1.00) CYP19A1ALDH1A1TSHRKIF11TRPV6
Triphenylmethanol SCHEMBL700 0.84 CYP19A1 (0.50) CYP19A1ALDH1A1TSHRCYP3A4CYP2D6
Triphenylmethanol SCHEMBL456603 0.84 CYP19A1 (0.50) CYP19A1ALDH1A1TSHRCYP3A4CYP2D6
Trifluoromethylbenzene SCHEMBL8692 0.84 TSHR (1.00) CYP19A1ALDH1A1TSHRKIF11TRPV6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8026263-B2 Methods for inhibiting neoproliferative changes in blood vessel walls THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2011-09-27 US disclosed
US-8026263-B2 Methods for inhibiting neoproliferative changes in blood vessel walls THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2011-09-27 US disclosed
US-7531573-B2 potent, selective and safe inhibitors of the Ca2+-activated potassium channel CHILDREN'S MEDICAL CENTER CORPORATION (US) 2009-05-12 US disclosed
US-7531573-B2 potent, selective and safe inhibitors of the Ca2+-activated potassium channel CHILDREN'S MEDICAL CENTER CORPORATION (US) 2009-05-12 US disclosed
US-7235577-B1 Non-peptide inhibition of T-lymphocyte activation and therapies related thereto THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2007-06-26 US disclosed
US-7235577-B1 Non-peptide inhibition of T-lymphocyte activation and therapies related thereto THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2007-06-26 US disclosed