SCHEMBL12296386

SCHEMBL12296386

CNC(C)c1cccc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.49
DAO P14920 1/20 0.47
IDO1 P14902 1/20 0.46
TDO2 P48775 1/20 0.46
SOS1 Q07889 2/20 0.46
HTR2A P28223 2/20 0.46
HTR2B P41595 2/20 0.46
HTR2C P28335 1/20 0.46
KRAS P01116 1/20 0.45
CES2 O00748 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
ACP3 P15309 1/20 0.45
LMNA P02545 2/20 0.45
MEN1 O00255 1/20 0.45
POLB P06746 1/20 0.45
HTT P42858 1/20 0.45
KMT2A Q03164 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
SLC6A4 P31645 2/20 0.44
SIGMAR1 Q99720 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10087246 1.00 PNMT (0.49) PNMTDAOIDO1TDO2SOS1
SCHEMBL8259841 1.00 PNMT (0.49) PNMTDAOIDO1TDO2SOS1
SCHEMBL17481894 0.85 PNMT (0.49) PNMTDAOIDO1TDO2SOS1
SCHEMBL25863567 0.84 PNMT (0.51) PNMTDAOIDO1TDO2SOS1
SCHEMBL10087175 0.84 NPSR1 (0.47) PNMTDAOIDO1TDO2SOS1
SCHEMBL29600944 0.83 CES2 (0.50) PNMTDAOIDO1TDO2HTR2A
SCHEMBL17465593 0.83 CES2 (0.50) PNMTDAOIDO1TDO2HTR2A
SCHEMBL4524501 0.83 CES2 (0.50) PNMTDAOIDO1TDO2HTR2A
SCHEMBL2538654 0.83 CES2 (0.50) PNMTDAOIDO1TDO2HTR2A
SCHEMBL6841423 0.82 DAO (0.46) PNMTDAOIDO1TDO2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2817312-B1 NOVEL NEUROKININ 1 RECEPTOR ANTAGONIST COMPOUNDS LEO PHARMA AS (DK) 2016-02-17 EP disclosed
US-9181259-B2 Substituted pyrrolo[1,2-a]piperazines and pyrrolo[1,2-a][1,4]diazepines as neurokinin 1 receptor antagonists LEO PHARMA A/S (DK) 2015-11-10 US disclosed
EP-2817312-A1 NOVEL NEUROKININ 1 RECEPTOR ANTAGONIST COMPOUNDS Leo Pharma A/S (DK) 2014-12-31 EP disclosed
WO-2013124286-A1 NOVEL NEUROKININ 1 RECEPTOR ANTAGONIST COMPOUNDS LEO PHARMA A/S (DK) 2013-08-29 WO disclosed
US-8470889-B2 Hybrid-ionone and curcumin molecules as anticancer agents TRT PHARMA INC. (CA) 2013-06-25 US disclosed
US-20110230488-A1 HYBRID-IONONE AND CURCUMIN MOLECULES AS ANTICANCER AGENTS TRT PHARMA INC. (CA) 2011-09-22 US disclosed
WO-2010060214-A1 HYBRID -IONONE AND CURCUMIN MOLECULES AS ANTICANCER AGENTS TRT PHARMA INC . (CA) 2010-06-03 WO disclosed
US-7713961-B2 Substituted 1,2-ethylenediamines, methods for preparing them and uses thereof BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-05-11 US disclosed
US-20090325940-A1 Substituted 1,2-ethylenediamines, Methods for Preparing Them and Uses Thereof BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-12-31 US disclosed
CN-100413850-C Chemical compounds GLAXO GROUP LTD (GB) 2008-08-27 CN disclosed
CN-1391564-A Chemical compounds GLAXO GROUP LTD (GB) 2003-01-15 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110230488-A1 HYBRID-IONONE AND CURCUMIN MOLECULES AS ANTICANCER AGENTS IKBKG, HSD17B11, IKBKE PNMT 4192/4885DAO 4736/4885IDO1 2269/4885
US-20090325940-A1 Substituted 1,2-ethylenediamines, Methods for Preparing Them and Uses Thereof PSEN1, PSEN2, BACE1 PNMT 49/4885DAO 93/4885IDO1 768/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.