SCHEMBL12320879

SCHEMBL12320879

O=C(c1ccc(-c2ccccc2)cc1)N1CCc2ncnc(N3CCC4OCCCC4C3)c2C1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.61
KCNK9 Q9NPC2 1/20 0.61
FASN P49327 3/20 0.44
MTHFD2 P13995 5/20 0.42
HTR2B P41595 2/20 0.38
CFTR P13569 1/20 0.38
P2RY12 Q9H244 1/20 0.38
TNK2 Q07912 2/20 0.37
HPGD P15428 1/20 0.37
MAPK1 P28482 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
SLC6A7 Q99884 1/20 0.37
LMNA P02545 1/20 0.36
TRPV1 Q8NER1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2442034 1.00 KCNK3 (0.61) KCNK3KCNK9FASNMTHFD2HTR2B
SCHEMBL2410232 0.79 KCNK3 (0.72) KCNK3KCNK9MTHFD2CFTRP2RY12
SCHEMBL2410478 0.78 KCNK3 (0.73) KCNK3KCNK9FASNMTHFD2HTR2B
SCHEMBL2471575 0.78 KCNK3 (0.65) KCNK3KCNK9MTHFD2CFTRP2RY12
SCHEMBL2407040 0.77 KCNK3 (0.87) KCNK3KCNK9FASNMTHFD2HTR2B
SCHEMBL2407042 0.76 KCNK3 (0.68) KCNK3KCNK9MTHFD2HTR2BCFTR
SCHEMBL2406138 0.76 KCNK3 (1.00) KCNK3KCNK9MTHFD2HTR2BCFTR
SCHEMBL30664070 0.76 KCNK3 (1.00) KCNK3KCNK9MTHFD2HTR2BCFTR
SCHEMBL12321174 0.76 KCNK3 (0.67) KCNK3KCNK9MTHFD2HTR2BCFTR
SCHEMBL2406140 0.75 KCNK3 (0.66) KCNK3KCNK9MTHFD2HTR2BCFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011103715-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed
WO-2011106276-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed