SCHEMBL2410232

SCHEMBL2410232

COC1CCN(c2ncnc3c2CN(C(=O)c2ccc(-c4ccccc4)cc2)CC3)CC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.72
KCNK9 Q9NPC2 1/20 0.72
MTHFD2 P13995 3/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
HPGD P15428 2/20 0.45
P2RY12 Q9H244 1/20 0.42
CFTR P13569 1/20 0.42
CDK4 P11802 3/20 0.42
CCND1 P24385 3/20 0.42
POLB P06746 2/20 0.41
TRPV1 Q8NER1 1/20 0.41
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
LMNA P02545 1/20 0.41
SCN1A P35498 1/20 0.40
SCN2A Q99250 1/20 0.40
SCN3A Q9NY46 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2471575 0.91 KCNK3 (0.65) KCNK3KCNK9MTHFD2MEN1KMT2A
SCHEMBL2410478 0.86 KCNK3 (0.73) KCNK3KCNK9MTHFD2MEN1KMT2A
SCHEMBL2407040 0.85 KCNK3 (0.87) KCNK3KCNK9MTHFD2MEN1KMT2A
SCHEMBL30664070 0.84 KCNK3 (1.00) KCNK3KCNK9MTHFD2MEN1KMT2A
SCHEMBL2406138 0.84 KCNK3 (1.00) KCNK3KCNK9MTHFD2MEN1KMT2A
SCHEMBL2407042 0.82 KCNK3 (0.68) KCNK3KCNK9MTHFD2MEN1KMT2A
SCHEMBL2406140 0.81 KCNK3 (0.66) KCNK3KCNK9MTHFD2MEN1KMT2A
SCHEMBL12321174 0.80 KCNK3 (0.67) KCNK3KCNK9MTHFD2P2RY12CFTR
SCHEMBL2442034 0.79 KCNK3 (0.61) KCNK3KCNK9MTHFD2HPGDP2RY12
SCHEMBL12320879 0.79 KCNK3 (0.61) KCNK3KCNK9MTHFD2HPGDP2RY12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011106276-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO claimed
WO-2011103715-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO claimed
WO-2011106276-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed
WO-2011103715-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed
WO-2011103715-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed