SCHEMBL2406138

SCHEMBL2406138

CCCC(=O)C1CCN(c2ncnc3c2CN(C(=O)c2ccc(-c4ccccc4)cc2)CC3)CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 1.00
KCNK9 Q9NPC2 1/20 1.00
P2RY12 Q9H244 4/20 0.46
MTHFD2 P13995 2/20 0.43
CFTR P13569 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
ALDH1A1 P00352 2/20 0.41
PTGDR Q13258 2/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.40
CYP2C9 P11712 2/20 0.40
PTGER2 P43116 1/20 0.40
CYP1A2 P05177 1/20 0.40
HSD17B10 Q99714 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
MEN1 O00255 2/20 0.39
HPGD P15428 1/20 0.39
TSHR P16473 1/20 0.39
KMT2A Q03164 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
POLB P06746 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30664070 1.00 KCNK3 (1.00) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL2407040 0.93 KCNK3 (0.87) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL2410478 0.85 KCNK3 (0.73) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL2410232 0.84 KCNK3 (0.72) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL2407042 0.81 KCNK3 (0.68) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL12321174 0.80 KCNK3 (0.67) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL2406140 0.79 KCNK3 (0.66) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL2407799 0.79 KCNK3 (0.65) KCNK3KCNK9POLBHTR2B
SCHEMBL2471575 0.79 KCNK3 (0.65) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL12320879 0.76 KCNK3 (0.61) KCNK3KCNK9P2RY12MTHFD2CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011106276-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed
WO-2011103715-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed
WO-2011103715-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed