SCHEMBL2406140

SCHEMBL2406140

O=CCCCC1CCN(c2ncnc3c2CN(C(=O)c2ccc(-c4ccccc4)cc2)CC3)CC1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.66
KCNK9 Q9NPC2 1/20 0.66
P2RY12 Q9H244 1/20 0.41
MTHFD2 P13995 4/20 0.40
CFTR P13569 1/20 0.39
HTR2B P41595 2/20 0.39
ALDH1A1 P00352 2/20 0.39
SLC6A7 Q99884 2/20 0.39
TSHR P16473 1/20 0.39
FAAH O00519 1/20 0.38
DRD2 P14416 1/20 0.38
HTR2A P28223 1/20 0.38
DRD3 P35462 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2407042 0.95 KCNK3 (0.68) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL2410478 0.81 KCNK3 (0.73) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL2407040 0.81 KCNK3 (0.87) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL2410232 0.81 KCNK3 (0.72) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL30664070 0.79 KCNK3 (1.00) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL2406138 0.79 KCNK3 (1.00) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL2471575 0.76 KCNK3 (0.65) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL12321174 0.76 KCNK3 (0.67) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL12320879 0.75 KCNK3 (0.61) KCNK3KCNK9P2RY12MTHFD2CFTR
SCHEMBL2442034 0.75 KCNK3 (0.61) KCNK3KCNK9P2RY12MTHFD2CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011103715-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed