SCHEMBL12326845

SCHEMBL12326845

CCc1cncc(-c2cc(C)c3cnccc3c2)c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 2/20 0.43
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38
CYP11B1 P15538 5/20 0.35
CYP11B2 P19099 5/20 0.35
TOP2A P11388 1/20 0.35
GPR55 Q9Y2T6 1/20 0.34
MAOA P21397 2/20 0.34
GRM4 Q14833 1/20 0.34
CLK2 P49760 1/20 0.34
CLK3 P49761 1/20 0.34
DYRK1A Q13627 1/20 0.34
WNT3A P56704 1/20 0.33
CYP19A1 P11511 1/20 0.33
KDM4E B2RXH2 1/20 0.33
POLB P06746 1/20 0.33
HTT P42858 1/20 0.33
RAD52 P43351 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19663000 0.80 MAOA (0.40) TOP2AMAOAGRM4WNT3ACYP19A1
SCHEMBL17691566 0.75 MAPK10 (0.49) AKT1CYP11B1TOP2AGRM4CYP19A1
SCHEMBL13177775 0.74 CYP1A1 (0.45) PRMT5WDR77CYP11B1CYP11B2GPR55
SCHEMBL12327333 0.73 PRKCZ (0.43) DYRK1A
SCHEMBL3701838 0.72 CYP1A2 (0.52) CYP11B1CYP11B2TOP2AMAOAGRM4
SCHEMBL16118323 0.72 CYP2A6 (0.56) CYP11B1CYP11B2DYRK1ACYP19A1KDM4E
SCHEMBL12326764 0.70 TNF (0.43) AKT1CYP11B1CYP11B2WNT3A
SCHEMBL18848330 0.70 MAOA (0.42) TOP2AMAOAGRM4CYP19A1KDM4E
SCHEMBL19663009 0.69 MAOA (0.39) TOP2AMAOAGRM4WNT3AKDM4E
SCHEMBL23045962 0.68 ABL1 (0.38) AKT1CYP11B1CYP11B2GRM4WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2366699-A1 8-SUBSTITUTED ISOQUINOLINE DERIVATIVE AND USE THEREOF Asahi Kasei Pharma Corporation (JP) 2011-09-21 EP disclosed