SCHEMBL12330147

SCHEMBL12330147

CC(NO)c1cccc(Cl)c1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
COASY Q13057 1/20 0.47
ACP3 P15309 1/20 0.43
ADRB2 P07550 1/20 0.43
ADRB1 P08588 1/20 0.43
ADRB3 P13945 1/20 0.43
SLC2A1 P11166 2/20 0.42
HPGD P15428 2/20 0.42
ALDH1A1 P00352 1/20 0.42
CASR P41180 2/20 0.42
GPR139 Q6DWJ6 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
TSHR P16473 1/20 0.40
PNMT P11086 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28277765 0.83 COASY (0.46) COASYACP3ADRB2ADRB1ADRB3
SCHEMBL15247597 0.83 COASY (0.46) COASYACP3ADRB2ADRB1ADRB3
SCHEMBL178548 0.82 COASY (0.44) COASYACP3ADRB2ADRB1ADRB3
SCHEMBL8246636 0.82 COASY (0.44) COASYACP3ADRB2ADRB1ADRB3
SCHEMBL11455315 0.80 PNMT (0.44) COASYACP3ADRB2ADRB1ADRB3
SCHEMBL25627915 0.80 CASR (0.48) COASYACP3ADRB2ADRB1ADRB3
SCHEMBL24176088 0.77 ADRB1 (0.44) COASYACP3ADRB2ADRB1ADRB3
SCHEMBL10087248 0.77 ADRB2 (0.44) COASYADRB2ADRB1ADRB3SLC2A1
SCHEMBL10087187 0.77 SLC6A2 (0.51) COASYACP3ADRB2ADRB1ADRB3
SCHEMBL14044305 0.77 CASR (0.46) COASYACP3ADRB2ADRB1ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364984-A1 Inhibitors of serine proteases VERTEX PHARMACEUTICALS INCORPORATED (US) 2011-09-14 EP disclosed