SCHEMBL1233119

SCHEMBL1233119

Nc1nc2cc(Br)ccc2c2c1nc1n2CCCNC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 4/20 0.40
PTGES O14684 1/20 0.36
ACHE P22303 1/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
BACE1 P56817 1/20 0.32
HRH3 Q9Y5N1 2/20 0.32
PDPK1 O15530 1/20 0.31
JAK2 O60674 1/20 0.31
KCNH2 Q12809 1/20 0.31
HTT P42858 1/20 0.30
NLRP3 Q96P20 1/20 0.30
NCF1 P14598 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1233918 0.93 HRH4 (0.42) HRH4PTGESACHETLR8TLR7
Hydrochloric Acid SCHEMBL1233122 0.82 TLR7 (0.40) ACHETLR8TLR7KCNH2HTT
SCHEMBL2684172 0.81 ALDH1A1 (0.39) HRH4PTGESACHETLR8TLR7
Hydrochloric Acid SCHEMBL1233327 0.77 MCHR1 (0.44)
SCHEMBL10123157 0.77 HRH4 (0.39) HRH4PTGESACHETLR8TLR7
SCHEMBL1232864 0.76 HRH4 (0.38) HRH4PTGESACHETLR8TLR7
Hydrochloric Acid SCHEMBL1233645 0.75 NCF1 (0.44) HRH4TLR8TLR7KCNH2HTT
SCHEMBL202167 0.74 PIK3CA (0.38) HRH4PTGESACHETLR8TLR7
SCHEMBL1232765 0.73 HRH4 (0.39) HRH4PTGESACHETLR8TLR7
Trifluoroacetic Acid SCHEMBL203340 0.73 KDM4E (0.37) HRH4PTGESACHETLR8TLR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7888349-B2 Piperazine, [1,4]Diazepane, [1,4]Diazocane, and [1,5]Diazocane fused imidazo ring compounds 3M INNOVATIVE PROPERTIES COMPANY (US) 2011-02-15 US disclosed
US-20070167476-A1 Piperazine, [1,4]Diazepane, [1,4]Diazocane, and [1,5]Diazocane fused imidazo ring compounds 3M INNOVATIVE PROPERTIES COMPANY 2007-07-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070167476-A1 Piperazine, [1,4]Diazepane, [1,4]Diazocane, and [1,5]Diazocane fused imidazo ring compounds IL4, IL2, IL5 HRH4 55/4885PTGES 500/4885ACHE 2235/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.