SCHEMBL123642

SCHEMBL123642

c1ccc2c3c(ccc2c1)NNCC3

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.41
ALDH1A1 P00352 3/20 0.41
CYP2A6 P11509 1/20 0.41
TSHR P16473 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KDM4E B2RXH2 2/20 0.39
CYP1A2 P05177 2/20 0.39
HPGD P15428 2/20 0.39
CYP2C19 P33261 2/20 0.39
GLA P06280 1/20 0.39
CYP2C9 P11712 1/20 0.39
SIRT1 Q96EB6 1/20 0.39
HPRT1 P00492 1/20 0.38
PTPN22 Q9Y2R2 1/20 0.36
HIF1A Q16665 1/20 0.35
CYP1B1 Q16678 1/20 0.35
HTT P42858 1/20 0.35
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35
NCOA1 Q15788 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7856090 0.91 ALDH1A1 (0.37) HSD17B10ALDH1A1CYP2A6TSHRTDP1
SCHEMBL31712991 0.89 HSD17B10 (0.38) HSD17B10ALDH1A1CYP2A6TSHRTDP1
SCHEMBL1159909 0.84 HSD17B10 (0.44) HSD17B10ALDH1A1CYP2A6TSHRTDP1
SCHEMBL582334 0.82 NOTUM (0.46) HSD17B10ALDH1A1CYP2A6TSHRTDP1
Hydrochloric Acid SCHEMBL8013061 0.81 NOTUM (0.44) HSD17B10ALDH1A1CYP2A6TSHRTDP1
Bromide SCHEMBL5406141 0.81 NOTUM (0.44) HSD17B10ALDH1A1CYP2A6TSHRTDP1
Bromide SCHEMBL8014734 0.81 NOTUM (0.44) HSD17B10ALDH1A1CYP2A6TSHRTDP1
Hydrochloric Acid SCHEMBL5396075 0.81 NOTUM (0.44) HSD17B10ALDH1A1CYP2A6TSHRTDP1
Iodide SCHEMBL5402073 0.81 NOTUM (0.44) HSD17B10ALDH1A1CYP2A6TSHRTDP1
SCHEMBL31712962 0.77 HSD17B10 (0.41) HSD17B10ALDH1A1CYP2A6TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9186349-B2 Diaza heterocyclic compounds for phototherapy MALLINCKRODT LLC (US) 2015-11-17 US disclosed
US-9186349-B2 Diaza heterocyclic compounds for phototherapy MALLINCKRODT LLC (US) 2015-11-17 US disclosed
US-20120058954-A1 Diaza Heterocyclic Compounds for Phototherapy OCERA THERAPEUTICS LLC 2012-03-08 US disclosed
US-20120058954-A1 Diaza Heterocyclic Compounds for Phototherapy OCERA THERAPEUTICS LLC 2012-03-08 US disclosed
WO-2010132554-A2 DIAZA HETEROCYCLIC COMPOUNDS FOR PHOTOTHERAPY MALLINCKRODT INC. (US) 2010-11-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120058954-A1 Diaza Heterocyclic Compounds for Phototherapy BAD, BID, CASP3 HSD17B10 3325/4885ALDH1A1 544/4885CYP2A6 1928/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.