SCHEMBL12366144

SCHEMBL12366144

[C-]#[N+]CC(=O)NCc1ccc(Oc2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.54
MAPK14 Q16539 3/20 0.53
KMT2A Q03164 3/20 0.51
NPC1 O15118 2/20 0.50
LMNA P02545 1/20 0.50
CYP3A4 P08684 1/20 0.50
HTT P42858 1/20 0.50
MMP13 P45452 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
RECQL P46063 2/20 0.49
TSHR P16473 1/20 0.49
HRH3 Q9Y5N1 1/20 0.47
FFAR1 O14842 2/20 0.47
ERCC1 P07992 1/20 0.47
ERCC4 Q92889 1/20 0.47
FFAR4 Q5NUL3 1/20 0.47
MEN1 O00255 2/20 0.47
POLB P06746 1/20 0.47
GAA P10253 1/20 0.47
EPHX2 P34913 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11591975 0.86 GAA (0.59) HPGDKMT2ALMNACYP3A4HTT
SCHEMBL12366121 0.83 LMNA (0.64) KMT2ALMNASMN1; SMN2MEN1GAA
SCHEMBL13192876 0.83 HPGD (0.62) HPGDMAPK14KMT2ANPC1LMNA
SCHEMBL13192880 0.80 RNF4 (0.62) HPGDMAPK14KMT2ANPC1LMNA
SCHEMBL14944099 0.80 MAPK14 (0.61) HPGDMAPK14KMT2ANPC1LMNA
SCHEMBL10133183 0.80 NPC1 (0.75) HPGDMAPK14KMT2ANPC1LMNA
SCHEMBL1728537 0.79 MAPK14 (0.68) HPGDMAPK14KMT2ALMNACYP3A4
SCHEMBL18376355 0.79 TSHR (0.59) HPGDMAPK14KMT2ANPC1LMNA
SCHEMBL12366146 0.78 EPHX2 (0.53) CYP3A4SMN1; SMN2HRH3EPHX2PPARG
SCHEMBL22560078 0.78 CYP3A4 (0.66) HPGDMAPK14KMT2ANPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US disclosed