SCHEMBL12409490

SCHEMBL12409490

Cc1cnc(NCc2ccncc2)c2ncc(-c3ccc(O)cc3)n12

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FYN P06241 5/20 0.42
PIM1 P11309 2/20 0.39
POLB P06746 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
MKNK1 Q9BUB5 1/20 0.38
ADORA3 P0DMS8 2/20 0.37
IKBKB O14920 2/20 0.37
CHUK O15111 2/20 0.37
TTK P33981 2/20 0.37
ADRA2C P18825 1/20 0.36
FLT1 P17948 1/20 0.36
F2 P00734 1/20 0.36
CCNB2 O95067 1/20 0.35
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35
CCNB3 Q8WWL7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12409487 0.84 PTGS2 (0.45) FYNPIM1
SCHEMBL2177585 0.83 CA1 (0.48)
SCHEMBL12409243 0.79 TTK (0.57) FYNADORA3TTK
SCHEMBL12409489 0.78 NTRK1 (0.43) IKBKBCHUK
SCHEMBL12409494 0.78 FYN (0.43) FYNPIM1MKNK1ADORA3TTK
SCHEMBL12409282 0.73 TTK (0.55) POLBL3MBTL1ADORA3TTK
SCHEMBL12409486 0.72 CA1 (0.39) FYN
SCHEMBL12409483 0.71 PI4KB (0.44) CDK1
SCHEMBL8239625 0.70 ADORA3 (0.56) POLBL3MBTL1ADORA3TTKADRA2C
SCHEMBL12409327 0.70 FYN (0.47) FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2567960-A2 Imidazo[1,2-a]pyrazine compounds for treatment of viral infections such as hepatitis Biofocus DPI Limited (GB) 2013-03-13 EP disclosed
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-8362018-B2 Substituted imidazo[1,2-a]pyrazine compounds useful for the treatment of viral infections BIOFOCUS DPI, LTD. (GB) 2013-01-29 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS BIOFOCUS DPI, LTD. (GB) 2011-07-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110166147-A1 IMIDAZOPYRAZINE COMPOUNDS CYP3A5, HAVCR2, CYP3A43 FYN 3511/4885PIM1 429/4885POLB 1195/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.